SCHEMBL2579176

SCHEMBL2579176

CC(CCc1ccccc1)NC(=O)c1noc2c1CN(S(=O)(=O)c1ccc(OC(F)(F)F)cc1)CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.41
SCN9A Q15858 2/20 0.40
ALDH1A1 P00352 6/20 0.39
EGLN1 Q9GZT9 1/20 0.38
CTSL P07711 2/20 0.38
CTSS P25774 2/20 0.38
CTSK P43235 2/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
USP2 O75604 1/20 0.38
MAPT P10636 1/20 0.38
LIPE Q05469 1/20 0.38
HTT P42858 2/20 0.37
SCN3A Q9NY46 1/20 0.37
EPHX2 P34913 1/20 0.37
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2587146 0.88 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1EGLN1CTSSMEN1
SCHEMBL2583662 0.80 BCHE (0.47) EPHX2
SCHEMBL4260241 0.80 SMN1; SMN2 (0.46) SMN1; SMN2SCN9AEGLN1MEN1KMT2A
SCHEMBL2586748 0.78 GAA (0.41) SMN1; SMN2ALDH1A1EGLN1MEN1KMT2A
SCHEMBL2579157 0.77 SMN1; SMN2 (0.42) SMN1; SMN2ALDH1A1EGLN1MEN1KMT2A
SCHEMBL15300377 0.75 CRHBP (0.39) MEN1KMT2ALIPEEPHX2
SCHEMBL2582491 0.74 ALDH1A1 (0.48) SMN1; SMN2ALDH1A1MEN1KMT2AUSP2
SCHEMBL2578768 0.74 TRPV1 (0.42) SMN1; SMN2ALDH1A1EGLN1KMT2AMAPT
SCHEMBL5531317 0.74 AKR1C3 (0.43) SMN1; SMN2SCN9AEGLN1MEN1KMT2A
SCHEMBL2578684 0.71 KDM4E (0.42) SMN1; SMN2ALDH1A1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed