SCHEMBL2583662

SCHEMBL2583662

O=C(NC1CCN(Cc2ccccc2)C1)c1noc2c1CN(S(=O)(=O)c1ccc(OC(F)(F)F)cc1)CC2

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.47
ACHE P22303 2/20 0.47
BACE1 P56817 2/20 0.47
DRD4 P21917 3/20 0.46
HTR2A P28223 2/20 0.46
CHRM4 P08173 7/20 0.46
CHRM2 P08172 5/20 0.46
CHRM1 P11229 3/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
DRD2 P14416 2/20 0.45
CCR2 P41597 1/20 0.45
EPHX2 P34913 1/20 0.44
CHRM5 P08912 2/20 0.43
CHRM3 P20309 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581672 0.88 DRD4 (0.53) BCHEACHEBACE1DRD4HTR2A
SCHEMBL2585658 0.84 CCR2 (0.46) DRD4HTR2AHDAC3HDAC4HDAC7
SCHEMBL2586918 0.84 CCR3 (0.51)
SCHEMBL2587146 0.81 SMN1; SMN2 (0.43) HDAC3HDAC4HDAC7HDAC9HDAC5
SCHEMBL2579176 0.80 SMN1; SMN2 (0.41) EPHX2
SCHEMBL2585643 0.79 MEN1 (0.43)
SCHEMBL4260241 0.79 SMN1; SMN2 (0.46) HDAC3HDAC4HDAC7HDAC9HDAC5
SCHEMBL2586748 0.76 GAA (0.41) EPHX2
SCHEMBL2579157 0.75 SMN1; SMN2 (0.42) HDAC3HDAC4HDAC7HDAC9HDAC5
SCHEMBL5531317 0.72 AKR1C3 (0.43) HDAC3HDAC4HDAC7HDAC9HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed