SCHEMBL2581672

SCHEMBL2581672

O=C(NC1CCN(Cc2ccc(C(F)(F)F)cc2)C1)c1noc2c1CN(S(=O)(=O)c1ccccc1)CC2

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.53
DRD2 P14416 4/20 0.53
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
NCOR2 Q9Y618 1/20 0.49
HTR2A P28223 2/20 0.47
TEAD1 P28347 1/20 0.47
SIGMAR1 Q99720 2/20 0.45
CCR2 P41597 3/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
BACE1 P56817 1/20 0.45
SLC6A5 Q9Y345 1/20 0.44
LMNA P02545 1/20 0.44
CHRM4 P08173 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2585658 0.93 CCR2 (0.46) DRD4DRD2HDAC3HDAC4HDAC7
SCHEMBL2583662 0.88 BCHE (0.47) DRD4DRD2HDAC3HDAC4HDAC7
SCHEMBL2586918 0.87 CCR3 (0.51) SIGMAR1
SCHEMBL2585643 0.79 MEN1 (0.43) LMNA
SCHEMBL2585178 0.73 ALDH1A1 (0.47) LMNA
SCHEMBL2585594 0.72 ALDH1A1 (0.49) LMNA
SCHEMBL2582295 0.72 GAA (0.42) LMNA
SCHEMBL2582036 0.72 GAA (0.52) LMNA
SCHEMBL4264547 0.71 KMT2A (0.48)
SCHEMBL2580912 0.71 TEAD1 (0.54) DRD4DRD2HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed