SCHEMBL2581684

SCHEMBL2581684

O=C(c1noc2ccncc12)N(CCc1ccccc1)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.46
RCE1 Q9Y256 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
DAGLA Q9Y4D2 1/20 0.41
LIMK1 P53667 1/20 0.40
LIMK2 P53671 1/20 0.40
C5AR1 P21730 1/20 0.40
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 1/20 0.39
MAPT P10636 1/20 0.39
LPAR1 Q92633 1/20 0.39
LPAR5 Q9H1C0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2589522 0.76 EPHX2 (0.56) KMT2AMEN1MAPTL3MBTL1KDM6B
SCHEMBL2585707 0.75 RAB9A (0.54) CYP1A2CYP2D6CYP2C9CYP2C19KMT2A
SCHEMBL3054586 0.75 RCE1 (0.60) PIN1RCE1CYP1A2CYP3A4CYP2D6
SCHEMBL2585532 0.72 HIF1A (0.52) CYP1A2CYP2D6CYP2C19KMT2AROCK1
SCHEMBL28072874 0.72 POLB (0.56) PIN1RCE1CYP1A2CYP3A4CYP2D6
SCHEMBL15111089 0.70 RCE1 (0.68) RCE1KMT2AMEN1LIMK1LIMK2
SCHEMBL2586922 0.68 HIF1A (0.72) ROCK1NPC1RAB9A
SCHEMBL7228409 0.68 MEN1 (0.61) RCE1KMT2AMEN1LIMK1LIMK2
SCHEMBL7553695 0.68 KDM4E (0.57) PIN1RCE1KMT2AMEN1C5AR1
SCHEMBL4062630 0.67 PIN1 (0.49) PIN1RCE1KMT2AMEN1LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed