SCHEMBL25825837

SCHEMBL25825837

CC(=O)c1ccc2c(c1O)CC1(C2)CN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.40
NR1H2 P55055 2/20 0.37
GPR119 Q8TDV5 2/20 0.36
OXTR P30559 1/20 0.36
AVPR1A P37288 1/20 0.36
CYP11B2 P19099 1/20 0.35
GPR183 P32249 1/20 0.35
MAPK1 P28482 1/20 0.34
SCD5 Q86SK9 1/20 0.34
HDAC1 Q13547 1/20 0.34
SPR P35270 2/20 0.34
DDB1 Q16531 2/20 0.34
CRBN Q96SW2 2/20 0.34
POLB P06746 1/20 0.33
ACACB O00763 1/20 0.33
PARP1 P09874 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25825838 0.82 ESR2 (0.35) ESR2NR1H2GPR119GPR183HDAC1
SCHEMBL25825836 0.80 ESR1 (0.36) ESR2MAPK1
SCHEMBL25825899 0.80 ESR2 (0.49) ESR2NR1H2GPR119MAPK1HDAC1
SCHEMBL25604351 0.78 ESR2 (0.53) ESR2NR1H2GPR119MAPK1POLB
SCHEMBL21940889 0.77 MAPK1 (0.50) ESR2NR1H2GPR119CYP11B2GPR183
SCHEMBL29609197 0.77 MAPK1 (0.50) ESR2NR1H2GPR119CYP11B2GPR183
SCHEMBL25604259 0.77 ESR2 (0.58) ESR2NR1H2GPR119MAPK1HDAC1
SCHEMBL25604196 0.77 ESR2 (0.58) ESR2NR1H2GPR119MAPK1HDAC1
SCHEMBL23051565 0.74 SCD5 (0.40) ESR2NR1H2GPR119OXTRAVPR1A
SCHEMBL23051561 0.72 GPR119 (0.41) ESR2NR1H2GPR119OXTRAVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed