SCHEMBL25825939

SCHEMBL25825939

COc1cc2c(cc1C)CN(Cc1ccccc1)C2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REV1 Q9UBZ9 1/20 0.55
SIGMAR1 Q99720 3/20 0.54
HTR1A P08908 1/20 0.54
ADRA2A P08913 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
DRD4 P21917 1/20 0.54
SLC6A2 P23975 1/20 0.54
HTR2C P28335 1/20 0.54
SLC6A4 P31645 1/20 0.54
OPRK1 P41145 1/20 0.54
HTR2B P41595 1/20 0.54
HTR5A P47898 1/20 0.54
SLC6A3 Q01959 1/20 0.54
TMEM97 Q5BJF2 1/20 0.54
KMT2A Q03164 3/20 0.50
BCHE P06276 2/20 0.50
MAPT P10636 3/20 0.48
ALDH1A1 P00352 2/20 0.48
ABCB1 P08183 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3051745 0.91 REV1 (0.64) REV1SIGMAR1HTR1AADRA2AADRA2B
SCHEMBL8793776 0.82 REV1 (0.70) REV1SIGMAR1HTR1AADRA2AADRA2B
SCHEMBL18356020 0.78 SIGMAR1 (0.51) REV1SIGMAR1HTR1AADRA2AADRA2B
SCHEMBL30073105 0.78 SIGMAR1 (0.60) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL3693352 0.77 SIGMAR1 (0.75) REV1SIGMAR1HTR1AADRA2AADRA2B
SCHEMBL10383284 0.76 ABCB1 (0.74) REV1SIGMAR1HTR1AADRA2AADRA2B
SCHEMBL5449836 0.76 HTR1A (0.54) REV1SIGMAR1HTR1AADRA2AADRA2B
SCHEMBL13726504 0.76 CRHBP (0.69) SIGMAR1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL3051392 0.75 CA2 (0.73) REV1DRD4TMEM97KMT2AMAPT
SCHEMBL3506177 0.75 CA2 (0.73) REV1DRD4TMEM97KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed