SCHEMBL25837978

SCHEMBL25837978

Cc1cc2c(c([C@@H]3CCCN3)c1)CCN(c1ccnn1C)C2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CHRM1 P11229 3/20 0.31
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
MAOA P21397 1/20 0.31
DRD1 P21728 1/20 0.31
SLC6A2 P23975 1/20 0.31
TEAD1 P28347 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
KCNH2 Q12809 1/20 0.31
TEAD4 Q15561 1/20 0.31
TEAD2 Q15562 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25838280 0.80 CREBBP (0.32) HSD17B10
SCHEMBL25303478 0.80 MAP3K12 (0.35) CYP1A2CYP3A4CYP2D6
SCHEMBL30068677 0.80 MAP3K12 (0.35) CYP1A2CYP3A4CYP2D6
SCHEMBL25303476 0.80 MAP3K12 (0.35) CYP1A2CYP3A4CYP2D6
SCHEMBL25838282 0.74 HSD17B10 (0.31) HSD17B10
SCHEMBL25838495 0.72 KCNH2 (0.33) HSD17B10MEN1KMT2ACHRM1KDM4E
SCHEMBL25838493 0.72 CHRNB2 (0.33) HSD17B10MEN1KMT2ACHRM1KDM4E
SCHEMBL25838310 0.71 MEN1 (0.35) MEN1KMT2ACHRM2CHRM4
SCHEMBL25837980 0.70 HSD17B10 (0.33) HSD17B10MEN1KMT2ACHRM1KDM4E
SCHEMBL25838497 0.70 THRB (0.33) HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed