SCHEMBL25859018

SCHEMBL25859018

CC#Cc1ccc(-c2nnc(N)nc2C)c(OCOCC)c1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.34
TSHR P16473 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
KMT2A Q03164 1/20 0.30
ATM Q13315 1/20 0.30
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25857680 0.88 S1PR1 (0.36) CACNA2D1TSHR
SCHEMBL31314251 0.88 CACNA2D1 (0.33) CACNA2D1TSHRGABRG2GABRB3GABRA5
SCHEMBL25859156 0.87 CHRNB2 (0.37) CACNA2D1TSHR
SCHEMBL25857483 0.80 ALOX5AP (0.43) ADORA2AADORA1ATM
SCHEMBL31314385 0.80 DHFR (0.40) CACNA2D1TSHR
SCHEMBL25857437 0.80 DHFR (0.40) CACNA2D1TSHR
SCHEMBL31314375 0.80 ALOX5AP (0.43) ADORA2AADORA1ATM
SCHEMBL25859255 0.79 CYP1A1 (0.33) CACNA2D1KMT2A
SCHEMBL25857924 0.77 CACNA2D1 (0.32) CACNA2D1GABRA1GABRG2GABRB3GABRA5
SCHEMBL25859817 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed