SCHEMBL25870686

SCHEMBL25870686

CCC(C)(C)C(=O)N1CCC2(CC1)CCN(c1ncc(C(=O)NC(C)C)cn1)CC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
USP2 O75604 3/20 0.39
CYP2D6 P10635 2/20 0.39
HIF1A Q16665 1/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
CYP2C9 P11712 5/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
CHRM4 P08173 1/20 0.38
JAK3 P52333 1/20 0.38
TIPARP Q7Z3E1 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
ALDH1A1 P00352 2/20 0.37
ACACB O00763 2/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25876576 0.91 CYP3A4 (0.43) CYP3A4MEN1KMT2AUSP2CYP2D6
SCHEMBL25876321 0.85 CYP3A4 (0.43) CYP3A4MEN1KMT2AUSP2CYP2D6
SCHEMBL25870687 0.77 CYP3A4 (0.41) CYP3A4MEN1KMT2AUSP2CYP2D6
SCHEMBL25870685 0.74 HIF1A (0.39) CYP3A4MEN1KMT2AUSP2CYP2D6
SCHEMBL5280671 0.74 MAPT (0.54) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL25870428 0.74 MEN1 (0.44) CYP3A4MEN1KMT2AUSP2CYP2D6
SCHEMBL25703284 0.70 HDAC3 (0.49) HDAC1HDAC3HDAC2HDAC8CHRM4
SCHEMBL12723192 0.70 CYP3A4 (0.48) CYP3A4MEN1KMT2ACYP2C9ALDH1A1
SCHEMBL12761286 0.67 HDAC3 (0.51) CYP3A4MEN1KMT2AHDAC1HDAC3
SCHEMBL28614518 0.67 CYP11B2 (0.51) CYP3A4ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116920-A1 PENTA- FUSED HEXA-HETEROCYCLIC COMPOUND, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE 杭州多域生物技术有限公司 2023-06-29 WO disclosed