Water

Water

SCHEMBL2587823

O.O.O.O.O=[N+]([O-])[O-].O=[N+]([O-])[O-].O=[N+]([O-])[O-].[Sc+3]

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
CA5A P35218 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
TSHR P16473 3/20 0.39
ALDH1A1 P00352 3/20 0.39
TDP1 Q9NUW8 1/20 0.39
HPGD P15428 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL8102707 1.00 MEN1 (0.67) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL16430834 1.00 MEN1 (0.67) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL3597571 1.00 MEN1 (0.67) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL2019827 1.00 MEN1 (0.67) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL2590832 0.94 MEN1 (0.75) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL28398822 0.94 MEN1 (0.75) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL10566608 0.94 MEN1 (0.75) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL28478211 0.94 MEN1 (0.75) MEN1KMT2ACA5ACA5BTSHR
SCHEMBL887970 0.94 MEN1 (0.75) MEN1KMT2ACA5ACA5BTSHR
Water SCHEMBL708617 0.94 MEN1 (0.75) MEN1KMT2ACA5ACA5BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806178-B1 CATALYST COMPOSED OF COMPLEX OXIDE ASAHI CHEMICAL IND (JP) 2020-03-04 EP disclosed
US-8642501-B2 Composite oxide catalyst ASAHI KASEI CHEMICALS CORPORATION (JP) 2014-02-04 US disclosed
US-8389435-B2 Metal oxide catalyst carrier particle and exhaust gas purification catalyst TOYOTA JIDOSHA KABUSHIKI KAISHA (JP) 2013-03-05 US disclosed
WO-2011135785-A1 PROPYLENE PRODUCTION METHOD TOYOTA JIDOSHA KABUSHIKI KAISHA (JP) 2011-11-03 WO disclosed
CN-101005892-B Catalyst composed of complex oxide ASAHI CHEMICAL CORP 2010-06-09 CN disclosed
US-20100004117-A1 METAL OXIDE CATALYST CARRIER PARTICLE AND EXHAUST GAS PURIFICATION CATALYST TOYOTA JIDOSHA KABUSHIKI KAISHA (JP) 2010-01-07 US disclosed
CN-101366139-A Electrolyte membrane, membrane electrode assembly, and fuel cell TOSHIBA KK (JP) 2009-02-11 CN disclosed
EP-2010319-A2 METAL OXIDE CATALYST CARRIER PARTICLE AND EXHAUST GAS PURIFICATION CATALYST Toyota Jidosha Kabushiki Kaisha (JP) 2009-01-07 EP disclosed
US-20080108843-A1 Composite Oxide Catalyst ASAHI KASEI CHEMICALS CORPORATION (JP) 2008-05-08 US disclosed
WO-2007113674-A2 METAL OXIDE CATALYST CARRIER PARTICLE AND EXHAUST GAS PURIFICATION CATALYST TOYOTA JIDOSHA KABUSHIKI KAISHA (GB) 2007-10-11 WO disclosed
CN-1344190-A Method for producing fine powder of metallic nickel comprised of fine spherical particles SAKAI CHEMICAL INDUSTRY CO (JP) 2002-04-10 CN disclosed
EP-1160033-A1 METHOD FOR PRODUCING FINE POWDER OF METALLIC NICKEL COMPRISED OF FINE SPHERICAL PARTICLES SAKAI CHEMICAL INDUSTRIAL COMPANY LTD. (JP) 2001-12-05 EP disclosed
EP-0658552-B1 Process for the preparation of alpha-tocopherol derivatives EISAI CO LTD (JP) 1999-03-31 EP disclosed
US-5532387-A CYCLIZATION OF TRIMETHYLHYDROQUINONE AND AN ALKENYL ALCOHOL, REUSABLE CATALYST, IIIB FLUOROSULFONATE, NITRATE, SULFATE, OR FLUOROALKYLSULFONATE EISAI CO., LTD. (JP) 1996-07-02 US disclosed
EP-0461850-B1 Process for producing alpha-hydroxycarboxylicacid amides MITSUI TOATSU CHEMICALS (JP) 1995-09-27 EP disclosed
EP-0658552-A1 Process for the preparation of alpha-tocopherol derivatives Eisai Co., Ltd. (JP) 1995-06-21 EP disclosed
US-5276185-A Reacting alpha hydroxy nitrile compound with water in presence of manganese dioxide catalyst containing a metal MITSUI TOATSU CHEMICALS, INC. (JP) 1994-01-04 US disclosed
US-5112783-A Containing chloride and/or nitrate, cubic structure UBE INDUSTRIES, LTD. (JP) 1992-05-12 US disclosed
EP-0461850-A1 Process for producing alpha-hydroxycarboxylicacid amides MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-12-18 EP disclosed
US-4003920-A OXIDATION OF UNSATURATED HYDROCARBONS KURARAY CO., LTD. (JA) 1977-01-18 US disclosed