SCHEMBL2588933

SCHEMBL2588933

CC(=O)On1nc(S(=O)(=O)Cc2ccccc2)c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 3/20 0.56
HCRTR1 O43613 2/20 0.56
MAPT P10636 4/20 0.40
POLB P06746 4/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HTR6 P50406 1/20 0.39
AGTR1 P30556 1/20 0.39
TSHR P16473 2/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TXNRD1 Q16881 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
MTOR P42345 1/20 0.36
HTT P42858 1/20 0.36
THRB P10828 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592911 0.88 HCRTR2 (0.54) HCRTR2HCRTR1MAPTPOLBKMT2A
SCHEMBL29092151 0.80 HCRTR1 (0.56) HCRTR2HCRTR1MAPTPOLBKMT2A
SCHEMBL7708626 0.76 HCRTR1 (0.71) HCRTR2HCRTR1MAPTPOLBKMT2A
SCHEMBL7708409 0.75 HCRTR1 (0.68) HCRTR2HCRTR1KMT2AMEN1ALDH1A1
SCHEMBL2596039 0.74 HCRTR1 (0.54) HCRTR2HCRTR1MAPTPOLBKMT2A
SCHEMBL2589420 0.72 HCRTR1 (0.39) HCRTR2HCRTR1MAPTPOLBKMT2A
SCHEMBL7704867 0.72 HCRTR2 (1.00) HCRTR2HCRTR1MAPTPOLBALDH1A1
SCHEMBL2592992 0.67 ATM (0.57) HCRTR2HCRTR1MAPTPOLBKMT2A
SCHEMBL498618 0.66 KMT2A (0.53) MAPTKMT2AALDH1A1TSHRHSD17B10
SCHEMBL2588315 0.66 L3MBTL1 (0.65) HCRTR2HCRTR1MAPTPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138265-A2 INDOLE AND INDAZOLE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed