SCHEMBL2594966

SCHEMBL2594966

Cc1ccc(C(=O)O)c(=O)[nH]1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.56
KDM4E B2RXH2 8/20 0.53
GAA P10253 5/20 0.52
HSD17B10 Q99714 3/20 0.52
HPGD P15428 2/20 0.52
ALDH1A1 P00352 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
NAPRT Q6XQN6 1/20 0.45
KDM3B Q7LBC6 1/20 0.42
CYP1A2 P05177 1/20 0.42
KDM6B O15054 1/20 0.42
KDM4A O75164 1/20 0.42
KDM4D Q6B0I6 1/20 0.42
HIF1AN Q9NWT6 1/20 0.42
KDM2A Q9Y2K7 1/20 0.42
HMBS P08397 1/20 0.42
NOTUM Q6P988 1/20 0.40
GLA P06280 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4513216 0.83 SPR (0.56) SPRKDM4EGAAHSD17B10HPGD
SCHEMBL5791701 0.81 SPR (0.54) SPRKDM4EGAAHSD17B10HPGD
Hydrochloric Acid SCHEMBL5010691 0.79 SPR (0.53) SPRKDM4EGAAHSD17B10HPGD
SCHEMBL4734537 0.78 KDM4E (0.68) SPRKDM4EGAAHSD17B10HPGD
SCHEMBL17770626 0.76 KDM4E (0.55) KDM4EGAAHSD17B10HPGDALDH1A1
SCHEMBL11120767 0.75 SPR (0.49) SPRKDM4EGAAHSD17B10HPGD
SCHEMBL8121938 0.75 ALDH1A1 (0.60) SPRKDM4EGAAALDH1A1GLA
SCHEMBL4230546 0.74 KDM4E (0.53) KDM4EGAAHSD17B10HPGDALDH1A1
SCHEMBL31547664 0.74 KDM4E (0.53) KDM4EGAAHSD17B10HPGDALDH1A1
SCHEMBL17503590 0.74 KDM4E (0.53) KDM4EGAAHSD17B10HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 93 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12466821-B2 Antiviral pyridopyrazinedione compounds NOVARTIS AG (CH) 2025-11-11 US disclosed
US-20240374583-A1 USE OF MORPHINAN DERIVATIVES FOR TREATMENT OF OPIOID DELTA RECEPTOR AGONIST-RELATED DISEASE NIPPON CHEMIPHAR CO., LTD (JP) 2024-11-14 US disclosed
US-12109209-B2 Use of morphinan derivatives for treatment of opioid delta receptor agonist-related disease NIPPON CHEMIPHAR CO., LTD. (JP) 2024-10-08 US disclosed
EP-4414037-A2 MORPHINAN DERIVATIVES FOR THE TREATMENT OF OPIOID DELTA RECEPTOR AGONIST-RELATED DISEASES Nippon Chemiphar Co., Ltd. (JP) 2024-08-14 EP disclosed
WO-2024158878-A1 FUSED TETRACYCLIC SELECTIVE PARP1 INHIBITORS ENLIVEN INC. (US) 2024-08-02 WO disclosed
EP-3513792-B9 MORPHINAN DERIVATIVES FOR THE TREATMENT OF OPIOID DELTA RECEPTOR AGONIST-RELATED DISEASES NIPPON CHEMIPHAR CO (JP) 2024-07-10 EP disclosed
WO-2024134514-A1 NOVEL COMPOUND AS RON INHIBITOR 주식회사 엘지화학 2024-06-27 WO disclosed
CN-113292559-B Morphinan derivatives 日本化学药品株式会社 2024-04-02 CN disclosed
EP-3513792-B1 MORPHINAN DERIVATIVES FOR THE TREATMENT OF OPIOID DELTA RECEPTOR AGONIST-RELATED DISEASES NIPPON CHEMIPHAR CO (JP) 2024-03-27 EP disclosed
US-20240018115-A1 ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE LOXO ONCOLOGY, INC. 2024-01-18 US disclosed
US-5312922-A Quinoline derivatives with hydroxy, trifluoromethyl, carboxy and/or bromo substituents NORDION INTERNATIONAL INC. (CA) 1994-05-17 US disclosed
EP-0509769-A2 Heterocyclic amides having HLE inhibiting activity ZENECA LIMITED (GB) 1992-10-21 EP disclosed
EP-0190265-B1 PYRIDONE ESTERS AS INOTROPIC AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-01-08 EP disclosed
EP-0190265-A4 PYRIDONE ESTERS AS INOTROPIC AGENTS. AMERICAN HOSPITAL SUPPLY CORP (US) 1987-07-09 EP disclosed
US-4657919-A CARDIOVASCULAR DISORDERS E. I. DU PONT DE NEMOURS & CO. (US) 1987-04-14 US disclosed
EP-0190265-A1 PYRIDONE ESTERS AS INOTROPIC AGENTS. AMERICAN HOSPITAL SUPPLY CORP (US) 1986-08-13 EP disclosed
WO-1986001202-A1 PYRIDONE ESTERS AS INOTROPIC AGENTS AMERICAN HOSPITAL SUPPLY CORPORATION (US) 1986-02-27 WO disclosed
US-4559347-A 3-Substituted-5-alkyl-1,6-naphthyridin-2(1H)-ones, cardiotonic use and preparation thereof STERLING DRUG INC. (US) 1985-12-17 US disclosed
US-4555517-A Pyridone esters as inotropic agents AMERICAN HOSPITAL SUPPLY CORPORATION (US) 1985-11-26 US disclosed
US-3965107-A Isothiazolopyridinones ROHM AND HAAS COMPANY (US) 1976-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240018115-A1 ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE PIK3CA, PIK3R4, PIK3R5 SPR 2629/4885KDM4E 2656/4885GAA 1962/4885
US-12466821-B2 Antiviral pyridopyrazinedione compounds ZC3HAV1, IL5, TYMP SPR 3931/4885KDM4E 508/4885GAA 1363/4885
US-20240374583-A1 USE OF MORPHINAN DERIVATIVES FOR TREATMENT OF OPIOID DELTA RECEPTOR AGONIST-RELATED DISEASE OPRD1, OPRM1, OPRK1 SPR 2233/4885KDM4E 4829/4885GAA 1826/4885
US-12109209-B2 Use of morphinan derivatives for treatment of opioid delta receptor agonist-related disease OPRD1, OPRM1, OPRK1 SPR 2233/4885KDM4E 4829/4885GAA 1826/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.