SCHEMBL2599705

SCHEMBL2599705

COc1ccc(Br)cc1O.CS(=O)(=O)O

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 known ✓ Q9H4B7 2/20 0.45
WDR5 P61964 5/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GLA P06280 1/20 0.50
MYC P01106 1/20 0.50
ALDH1A1 P00352 3/20 0.47
AOX1 Q06278 1/20 0.47
MAPT P10636 3/20 0.47
HSD17B10 Q99714 2/20 0.47
GFER P55789 1/20 0.47
TSHR P16473 1/20 0.46
ACLY P53396 1/20 0.46
LMNA P02545 2/20 0.46
GAA P10253 3/20 0.45
PTGS1 P23219 1/20 0.45
APP P05067 1/20 0.45
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
THRB P10828 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30152196 0.89 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1AOX1MAPTHSD17B10
SCHEMBL41497 0.89 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1AOX1MAPTHSD17B10
Formaldehyde SCHEMBL27568605 0.87 ALDH1A1 (0.52) WDR5SMN1; SMN2MYCALDH1A1AOX1
Bicarbonate SCHEMBL28501235 0.85 GAA (0.54) SMN1; SMN2ALDH1A1AOX1MAPTHSD17B10
SCHEMBL19509694 0.78 ALDH1A1 (0.45) WDR5SMN1; SMN2GLAMYCALDH1A1
SCHEMBL27584635 0.76 SMN1; SMN2 (0.59) WDR5SMN1; SMN2GLAMYCALDH1A1
SCHEMBL2123784 0.76 PTGS1 (0.57) SMN1; SMN2ALDH1A1AOX1MAPTHSD17B10
Hydrochloric Acid SCHEMBL27582675 0.75 SMN1; SMN2 (0.58) WDR5SMN1; SMN2GLAMYCALDH1A1
Sulfuric Acid SCHEMBL28214565 0.75 CA1 (0.53) SMN1; SMN2GLAALDH1A1MAPTTSHR
SCHEMBL1790129 0.74 SMN1; SMN2 (0.65) WDR5SMN1; SMN2GLAMYCALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2574192-B1 PROCESS FOR PREPARING AN ORTHO-SUBSTITUTED 5-HALOPHENOL AND A SYNTHESIS INTERMEDIATE THEREOF RHODIA CHINA CO LTD (CN) 2016-09-21 EP disclosed
US-8975431-B2 Process for preparing an ortho-substituted 5-halophenol and a synthesis intermediate thereof RHODIA OPERATIONS (FR) 2015-03-10 US disclosed
EP-2574192-A1 PROCESS FOR PREPARING AN ORTHO-SUBSTITUTED 5-HALOPHENOL AND A SYNTHESIS INTERMEDIATE THEREOF Rhodia (China) Co., Ltd. (CN) 2013-04-03 EP disclosed
US-20130066097-A1 PROCESS FOR PREPARING AN ORTHO-SUBSTITUTED 5-HALOPHENOL AND A SYNTHESIS INTERMEDIATE THEREOF RHODIA (CHINA) CO., LTD. (CN) 2013-03-14 US disclosed
WO-2011143819-A1 PROCESS FOR PREPARING AN ORTHO-SUBSTITUTED 5-HALOPHENOL AND A SYNTHESIS INTERMEDIATE THEREOF RHODIA (CHINA) CO., LTD. (CN) 2011-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130066097-A1 PROCESS FOR PREPARING AN ORTHO-SUBSTITUTED 5-HALOPHENOL AND A SYNTHESIS INTERMEDIATE THEREOF HDHD5, HPD, NISCH TUBB1 4726/4885WDR5 3551/4885SMN1; SMN2 4595/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.