SCHEMBL26046355

SCHEMBL26046355

COc1c(O)ccc(CCC(=O)O)c1CO

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.55
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
GAA P10253 1/20 0.39
FFAR4 Q5NUL3 2/20 0.38
ALDH1A1 P00352 1/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
FFAR1 O14842 1/20 0.37
IMPDH2 P12268 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
F2 P00734 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26046416 0.88 IAPP (0.45) POLBMAPTTP53TRPV1ALDH1A1
SCHEMBL26046360 0.86 POLB (0.47) POLBNPSR1GAAFFAR4ALDH1A1
SCHEMBL21317655 0.83 POLB (0.61) POLBNPSR1TRPV1GAAALDH1A1
SCHEMBL21317652 0.82 POLB (0.59) POLBNPSR1TRPV1GAAALDH1A1
SCHEMBL26046493 0.82 HMGCR (0.43) POLBTRPV1
SCHEMBL10748552 0.81 CA2 (0.39) POLBMAPTTRPV1GAAALDH1A1
SCHEMBL21317651 0.81 POLB (0.58) POLBNPSR1TRPV1GAAALDH1A1
SCHEMBL26046352 0.80 POLB (0.45) POLBNPSR1FFAR4ALDH1A1FFAR1
SCHEMBL26046358 0.80 POLB (0.50) POLBNPSR1MAPTGAAFFAR4
SCHEMBL16319477 0.76 POLB (0.55) POLBNPSR1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11746364-B2 Enzymatic synthesis of kavalactones and flavokavains WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2023-09-05 US disclosed
US-11739354-B2 Enzymatic synthesis of kavalactones and flavokavains WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2023-08-29 US disclosed