SCHEMBL26106532

SCHEMBL26106532

Cc1cc(F)c(B2OC(C)(C)C(C)(C)O2)c(C(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
CSNK2A1 P68400 1/20 0.35
NOTUM Q6P988 3/20 0.34
P4HB P07237 1/20 0.33
ROCK1 Q13464 1/20 0.33
F2 P00734 1/20 0.33
F11 P03951 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
PRSS3 P35030 1/20 0.33
METAP2 P50579 1/20 0.33
LPL P06858 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
TPMT P51580 1/20 0.32
DHODH Q02127 4/20 0.32
MYC P01106 1/20 0.32
TTR P02766 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PDGFRB P09619 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL327717 0.83 LPL (0.40) ROCK1LPLLIPG
SCHEMBL13125462 0.79 LMNA (0.38) KDM4EP4HBROCK1F2F11
SCHEMBL12470639 0.77 HSD17B10 (0.36) KDM4EALDH1A1
SCHEMBL16535080 0.75 CES2 (0.37) ROCK1F2F11PRSS1PRSS2
SCHEMBL13125464 0.75 ROCK1 (0.33) P4HBROCK1F2F11PRSS1
SCHEMBL23354375 0.75 CES2 (0.38) P4HBROCK1F2F11PRSS1
SCHEMBL17939966 0.74 ROCK1 (0.39) KDM4EP4HBROCK1F2F11
SCHEMBL10059440 0.74 RXRA (0.35) KDM4ENOTUMROCK1F2F11
SCHEMBL17873998 0.74 RXRA (0.35) KDM4ENOTUMP4HBROCK1F2
SCHEMBL17939981 0.74 LPL (0.35) KDM4EP4HBROCK1F2F11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023179600-A1 NOVEL SUBSTITUTED MACROHETEROCYCLIC COMPOUNDS AND USE THEREOF 杭州德睿智药科技有限公司 2023-09-28 WO disclosed