SCHEMBL2620993

SCHEMBL2620993

CCc1ccc2scnc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.47
RAB9A P51151 5/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 2/20 0.45
HSD17B10 Q99714 1/20 0.45
TRPM5 Q9NZQ8 1/20 0.40
FFAR1 O14842 1/20 0.40
RIPK2 O43353 2/20 0.39
LCK P06239 2/20 0.39
KDR P35968 2/20 0.39
TGFBR1 P36897 2/20 0.39
PTK6 Q13882 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
MAPK1 P28482 1/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
ESR1 P03372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6647512 0.85 ALDH1A1 (0.42) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL763958 0.85 NPC1 (0.57) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL29976332 0.82 ALDH1A1 (0.47) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9676880 0.82 ALDH1A1 (0.47) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9507208 0.82 SKP2 (0.41) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL27610684 0.81 CLK1 (0.42) NPC1RAB9ASMN1; SMN2ALDH1A1HSD17B10
SCHEMBL20621822 0.81 TRPM5 (0.42) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL13610284 0.81 ALDH1A1 (0.45) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL3819546 0.81 ALDH1A1 (0.45) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6396893 0.81 CYP2A6 (0.47) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 151 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4400504-A1 THIOPHENE RING COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Center for Excellence in Molecular Cell Science, Chinese Academy of Sciences (CN) 2024-07-17 EP disclosed
WO-2024059249-A1 M4 ACTIVATORS/MODULATORS AND USES THEREOF CEREVEL THERAPEUTICS, LLC (US) 2024-03-21 WO disclosed
US-20230382907-A1 5- AND 6-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES ENLIVEN INC. 2023-11-30 US disclosed
US-11807649-B2 Fused tetracyclic quinazoline derivatives as inhibitors of ErbB2 ENLIVEN THERAPEUTICS, INC. (US) 2023-11-07 US disclosed
US-11807638-B2 5- and 6-azaindole compounds for inhibition of Bcr-Abl tyrosine kinases ENLIVEN INC. (US) 2023-11-07 US disclosed
US-11767321-B2 5- and 6-azaindole compounds for inhibition of BCR-ABL tyrosine kinases ENLIVEN INC. (US) 2023-09-26 US disclosed
EP-3640248-B1 AMINOPYRIMIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND USE THEREOF BEIJING ADAMADLE BIOTECHNOLOGY LLC (CN) 2023-08-23 EP disclosed
WO-2023154124-A1 ACYLATED HETEROCYCLIC QUINAZOLINE DERIVATIVES AS INHIBITORS OF ERBB2 ENLIVEN THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed
EP-3582783-B1 7-MEMBERED AZA-HETEROCYCLIC CONTAINING DELTA-OPIOID RECEPTOR MODULATING COMPOUNDS, METHODS OF USING AND MAKING THE SAME TREVENA INC (US) 2023-06-07 EP disclosed
US-11661418-B2 MASP-2 inhibitors and methods of use OMEROS CORPORATION (US) 2023-05-30 US disclosed
US-4917997-A MIXED WITH ASCORBIC ACID COMPONENT, SENSITIZING DYE, BISAMINOSTILBENE WITH PYRIMIDINE SUBSTITUTION FUJI PHOTO FILM CO., LTD. (JP) 1990-04-17 US disclosed
US-4894321-A SILVER HALIDE EMULSIONS, IMAGES, MULTILAYER FUJI PHOTO FILM CO., LTD. (JP) 1990-01-16 US disclosed
EP-0331185-A2 Silver halide photographic element for forming direct positive images and a method for forming said images FUJI PHOTO FILM CO., LTD. (JP) 1989-09-06 EP disclosed
US-4851327-A THIN SOLID METAL FILM FUJI PHOTO FILM CO., LTD. (JP) 1989-07-25 US disclosed
EP-0316456-A1 ESTER-SUBSTITUTED THIENOTRIAZOLODIAZEPINE COMPOUNDS AND THEIR MEDICINAL USE Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-05-24 EP disclosed
US-4822726-A HIGH SILVER CHLORIDE CONCENTRATION FUJI PHOTO FILM CO., LTD. (JP) 1989-04-18 US disclosed
EP-0287100-A2 Silver halide photographic material FUJI PHOTO FILM CO., LTD. (JP) 1988-10-19 EP disclosed
EP-0253390-A2 Photographic support and color photosensitive material FUJI PHOTO FILM CO., LTD. (JP) 1988-01-20 EP disclosed
US-4010037-A Spectrally sensitized silver halide photographic emulsion FUJI PHOTO FILM CO., LTD. (JA) 1977-03-01 US disclosed
US-3966477-A Spectrally sensitized silver halide photographic emulsion FUJI PHOTO FILM CO., LTD. (JA) 1976-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11807638-B2 5- and 6-azaindole compounds for inhibition of Bcr-Abl tyrosine kinases ABL1, ABL2, BCR NPC1 4143/4885RAB9A 1191/4885SMN1; SMN2 3904/4885
US-20230382907-A1 5- AND 6-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES ABL1, ABL2, BCR NPC1 4143/4885RAB9A 1191/4885SMN1; SMN2 3904/4885
US-11767321-B2 5- and 6-azaindole compounds for inhibition of BCR-ABL tyrosine kinases ABL1, ABL2, BCR NPC1 4143/4885RAB9A 1191/4885SMN1; SMN2 3904/4885
US-11807649-B2 Fused tetracyclic quinazoline derivatives as inhibitors of ErbB2 ERBB2, ERBB3, BRCA1 NPC1 3640/4885RAB9A 1195/4885SMN1; SMN2 1701/4885
US-11661418-B2 MASP-2 inhibitors and methods of use MASP2, METAP2, SPINT2 NPC1 2354/4885RAB9A 2027/4885SMN1; SMN2 1476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.