SCHEMBL2632284

SCHEMBL2632284

CCOC(=O)c1ccc(O)o1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.60
HDAC6 Q9UBN7 1/20 0.60
ALDH1A1 P00352 8/20 0.54
MAPT P10636 4/20 0.54
KDM4E B2RXH2 3/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
TLR2 O60603 1/20 0.54
NSD2 O96028 1/20 0.54
POLB P06746 1/20 0.54
PKM P14618 1/20 0.54
MPI P34949 1/20 0.54
GRK6 P43250 1/20 0.54
RECQL P46063 1/20 0.54
TLR1 Q15399 1/20 0.54
TLR6 Q9Y2C9 1/20 0.54
LMNA P02545 2/20 0.51
CA12 O43570 4/20 0.48
CA1 P00915 4/20 0.48
CA2 P00918 4/20 0.48
CA7 P43166 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL449698 0.88 HDAC4 (0.73) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL29617026 0.84 HDAC4 (0.64) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL669793 0.82 HDAC4 (0.62) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL14052281 0.81 HDAC4 (0.70) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL1828976 0.81 HDAC4 (0.65) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL28427399 0.81 HDAC4 (0.65) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL22618595 0.80 ALDH1A1 (0.57) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL19287236 0.80 HDAC4 (0.42) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL362159 0.79 TSHR (0.63) HDAC4HDAC6ALDH1A1MAPTKDM4E
SCHEMBL3824966 0.79 HDAC4 (0.63) HDAC4HDAC6ALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158677-B2 Treatment of viral infections by modulation of host cell metabolic pathways THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2012-04-17 US disclosed
US-20090239830-A1 Treatment of viral infections by modulation of host cell metabolic pathways KADMON CORPORATION, LLC 2009-09-24 US disclosed
US-6465647-B1 Oxygen, sulfur and nitrogen substituted cyclohexene and cyclohexane derivatives having retinoid-like biological activity ALLERGAN, INC. 2002-10-15 US disclosed
US-6465646-B1 1-alkoxy and 1-acyloxy substituted cyclohex-1-ene compounds and sulfur and 1-alkoxycarbonyl analogs having retinoid-like biological activity ALLERGAN, INC. 2002-10-15 US disclosed
US-6177588-B1 HAVING RETINOID-LIKE, RETINOID ANTAGONIST OR RETINOID INVERSE AGONIST-LIKE BIOACTIVITY; SIDE EFFECT REDUCTION; SKIN DISORDERS; ANTIPROLIFERATIVE AND -CARCINOGENIC AGENTS; MICROBIOCIDES; VISION DEFECTS; CARDIOVASCULAR DISORDERS ALLERGAN SALES, INC. 2001-01-23 US disclosed
US-6166244-A Oxygen, sulfur and nitrogen substituted cyclohexene and cyclohexane derivatives having retinoid-like biological activity ALLERGAN SALES, INC. (US) 2000-12-26 US disclosed
WO-2000068191-A1 OXYGEN, SULFUR AND NITROGEN SUBSTITUTED CYCLOHEXENE AND CYCLOHEXANE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 2000-11-16 WO disclosed
WO-2000068190-A2 1-ALKOXY AND 1-ACYLOXY SUBSTITUTED CYCLOHEX-1-ENE COMPOUNDS AND SULFUR AND 1-ALKOXYCARBONYL ANALOGS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 2000-11-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090239830-A1 Treatment of viral infections by modulation of host cell metabolic pathways GOT2, MAVS, ME3 HDAC4 859/4885HDAC6 1725/4885ALDH1A1 1469/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.