SCHEMBL26465704

SCHEMBL26465704

CC(C)(C)NC(=O)CN1C2CC1CN(CC(=O)Nc1cc(F)cc(C#N)c1)C2

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 14/20 0.51
CACNA1G O43497 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
AR P10275 3/20 0.36
CYP2D6 P10635 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26465689 0.86 CACNA1H (0.54) CACNA1HCACNA1GCACNA1I
SCHEMBL26464490 0.85 CACNA1H (0.54) CACNA1HCACNA1GCACNA1ICYP2D6KCNH2
SCHEMBL26465573 0.83 CACNA1H (0.72) CACNA1H
SCHEMBL26465702 0.80 CACNA1H (0.43) CACNA1HAR
SCHEMBL26465838 0.79 CACNA1H (0.55) CACNA1HCACNA1GCACNA1ICYP2D6KCNH2
SCHEMBL26463608 0.79 CACNA1H (0.56) CACNA1HCACNA1GCACNA1ICYP2D6KCNH2
SCHEMBL26464783 0.78 CACNA1H (0.46) CACNA1HCACNA1GCACNA1ICYP2D6KCNH2
SCHEMBL26465699 0.77 HPGD (0.55) CACNA1HCYP2D6
SCHEMBL26465812 0.76 CACNA1H (0.47) CACNA1HCYP2D6
SCHEMBL26465810 0.76 CACNA1H (0.47) CACNA1HCACNA1GARCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192669-A1 T-TYPE CALCIUM CHANNEL MODULATORS COMPRISING A PIPERAZINE OR 1,4-DIAZEPANE CORE AND METHODS OF USE THEREOF PRAXIS PRECISION MEDICINES, INC. (US) 2023-10-05 WO disclosed