SCHEMBL2646586

SCHEMBL2646586

O=C(CNC(=O)c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1)Oc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 6/20 0.62
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
LMNA P02545 3/20 0.62
HTT P42858 2/20 0.62
MAPT P10636 2/20 0.62
PKM P14618 1/20 0.55
RAB9A P51151 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
ALDH1A1 P00352 2/20 0.50
FFAR1 O14842 1/20 0.48
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10424957 0.81 ALOX5 (0.67) ALOX5MEN1KMT2ALMNAHTT
SCHEMBL27554309 0.80 SMN1; SMN2 (0.56) HTTMAPTRAB9AALDH1A1GAA
SCHEMBL1134873 0.80 RAB9A (0.58) MEN1KMT2ALMNAHTTMAPT
SCHEMBL1578589 0.79 KMT2A (0.95) ALOX5MEN1KMT2ALMNAHTT
SCHEMBL28989406 0.78 MGLL (0.58) ALOX5MEN1KMT2AMAPTRAB9A
SCHEMBL28891518 0.78 SMN1; SMN2 (0.54) HTTMAPTRAB9AALDH1A1GAA
SCHEMBL11340446 0.78 PKM (0.56) ALOX5MEN1KMT2ALMNAHTT
SCHEMBL27182272 0.78 KMT2A (0.88) ALOX5MEN1KMT2ALMNAHTT
SCHEMBL455174 0.77 ALOX5 (0.72) ALOX5MEN1KMT2ALMNAHTT
SCHEMBL27935077 0.77 ALOX5 (1.00) ALOX5MEN1KMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255305-B1 PSYCHOLOGICAL DISORDERS MERCK SHARP & DOHME LIMITED (GB) 2001-07-03 US disclosed
EP-0915875-A2 SUBSTITUTED TRIAZOLO-PYRIDAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 1999-05-19 EP disclosed
WO-1998004559-A2 SUBSTITUTED TRIAZOLO-PYRIDAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1998-02-05 WO disclosed
US-5118690-A PHARMACEUTICAL TETRAHYDROISOQUINOLINES JOHN WYETH & BROTHER LIMITED (GB) 1992-06-02 US disclosed