SCHEMBL2646933

SCHEMBL2646933

COC(=O)c1cccc2c(Br)cccc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.57
MEN1 O00255 5/20 0.57
AHR P35869 1/20 0.57
PRNP P04156 1/20 0.53
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
ALDH1A1 P00352 2/20 0.47
CFTR P13569 1/20 0.47
HSD17B10 Q99714 1/20 0.47
SLC6A3 Q01959 1/20 0.46
BRD4 O60885 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46
CA9 Q16790 1/20 0.46
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.46
ATM Q13315 1/20 0.46
PSMD14 O00487 1/20 0.45
NR4A2 P43354 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29583255 1.00 KMT2A (0.57) KMT2AMEN1AHRPRNPLMNA
SCHEMBL869550 0.89 BRD4 (0.50) KMT2AMEN1AHRLMNATSHR
SCHEMBL70429 0.88 LMNA (0.59) KMT2AMEN1LMNATSHRALDH1A1
SCHEMBL25523280 0.86 SLC6A3 (0.56) KMT2AMEN1AHRPRNPLMNA
SCHEMBL30848483 0.85 PRNP (0.56) KMT2AMEN1AHRPRNPALDH1A1
SCHEMBL4959202 0.85 PRNP (0.56) KMT2AMEN1AHRPRNPALDH1A1
SCHEMBL31525357 0.82 KMT2A (0.45) KMT2AMEN1AHRPRNPLMNA
SCHEMBL29279663 0.81 TSHR (0.52) KMT2AMEN1LMNATSHRALDH1A1
SCHEMBL3230050 0.81 NR4A2 (0.53) LMNATSHRALDH1A1CFTRHSD17B10
SCHEMBL28485658 0.81 KMT2A (0.61) KMT2AMEN1AHRPRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3860636-B1 MATRIPTASE 2 INHIBITORS AND USES THEREOF DISC MEDICINE INC (US) 2026-01-28 EP disclosed
US-20250388593-A1 CEREBLON E3 LIGASE BINDING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND PRODUCTION METHOD THEREFOR MITSUBISHI TANABE PHARMA CORPORATION (JP) 2025-12-25 US disclosed
EP-4650348-A1 CEREBLON E3 LIGASE BINDING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND PRODUCTION METHOD THEREFOR Mitsubishi Tanabe Pharma Corporation (JP) 2025-11-19 EP disclosed
US-12428415-B2 Matriptase 2 inhibitors and uses thereof DISC MEDICINE, INC. (US) 2025-09-30 US disclosed
EP-4565121-A1 CARBON MONOXIDE PROBE MOLECULES Georgia State University Research Foundation, Inc. (US) 2025-06-11 EP disclosed
CN-119997870-A Carbon monoxide probe molecule 乔治亚州立大学研究基金会股份有限公司 2025-05-13 CN disclosed
US-12195472-B2 Substituted indole Mcl-1 inhibitors VANDERBILT UNIVERSITY (US) 2025-01-14 US disclosed
US-12144816-B2 Substituted indole Mcl-1 inhibitors VANDERBILT UNIVERSITY (US) 2024-11-19 US disclosed
WO-2024150815-A1 CEREBLON E3 LIGASE BINDING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND PRODUCTION METHOD THEREFOR 田辺三菱製薬株式会社 2024-07-18 WO disclosed
WO-2024030944-A1 CARBON MONOXIDE PROBE MOLECULES GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2024-02-08 WO disclosed
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
US-6495710-B2 Synthesis and use of dimethyl 1,5-naphthalenedicarboxlyates and intermediates therefrom BP CORPORATION NORTH AMERICA INC. 2002-12-17 US disclosed
US-20010031852-A1 Synthesis and use of dimethyl 1,5-naphthalenedicarboxylates and intermediates therefrom BP CORPORATION NORTH AMERICA INC. 2001-10-18 US disclosed
EP-1140823-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2001-10-10 EP disclosed
WO-2001051450-A2 SYNTHESIS AND USE OF DIMETHYL-1,5-NAPHTHALENEDICARBOXYLATES AND INTERMEDIATES THEREFROM BP CORPORATION NORTH AMERICA INC. (US) 2001-07-19 WO disclosed
US-6166034-A Spiro piperidine derivatives as 5HT1D receptor antagonists SMITHKLINE BEECHAM P. L. C (GB) 2000-12-26 US disclosed
WO-2000039088-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-07-06 WO disclosed
EP-0861257-A1 SPIRO PIPERIDINE DERIVATIVES AS 5MT RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-09-02 EP disclosed
WO-1997017351-A1 SPIRO PIPERIDINE DERIVATIVES AS 5MT RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-05-15 WO disclosed
US-5183825-A Antidiabetic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1993-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12428415-B2 Matriptase 2 inhibitors and uses thereof MMP7, MATR3, SPINT2 KMT2A 1072/4885MEN1 772/4885AHR 3258/4885
US-12144816-B2 Substituted indole Mcl-1 inhibitors MCL1, BCL2L1, BCL9 KMT2A 824/4885MEN1 3549/4885AHR 752/4885
US-20250388593-A1 CEREBLON E3 LIGASE BINDING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND PRODUCTION METHOD THEREFOR CRBN, CUL1, CBL KMT2A 663/4885MEN1 859/4885AHR 2566/4885
US-12195472-B2 Substituted indole Mcl-1 inhibitors MCL1, BCL2L1, BCL3 KMT2A 670/4885MEN1 2979/4885AHR 437/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.