SCHEMBL2649991

SCHEMBL2649991

CCOC(=O)C1C=NC(C)=C(c2ccc(Cl)cc2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
ALPL P05186 1/20 0.41
TARBP2 Q15633 1/20 0.41
MAPT P10636 3/20 0.41
PRKCZ Q05513 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
GABRA2 P47869 2/20 0.40
GABRB2 P47870 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GCGR P47871 1/20 0.40
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649546 0.87 HTT (0.44) LMNATARBP2MAPTNPSR1ALDH1A1
SCHEMBL2649211 0.87 RAB9A (0.43) LMNAMAPTNPSR1ALDH1A1MEN1
SCHEMBL2648348 0.86 ALDH1A1 (0.47) LMNATARBP2MAPTNPSR1ALDH1A1
SCHEMBL2651383 0.84 KDM4E (0.39) LMNAMAPTGABRA2NPSR1ALDH1A1
SCHEMBL2649285 0.83 RAB9A (0.48) LMNAMAPTPRKCZALDH1A1L3MBTL1
SCHEMBL2649878 0.76 ALDH1A1 (0.45) LMNAMAPTNPSR1ALDH1A1KMT2A
SCHEMBL2649623 0.76 CNR2 (0.43) CYP1A2
SCHEMBL2649291 0.75 MAPT (0.50) LMNAMAPTNPSR1ALDH1A1MEN1
SCHEMBL2649630 0.74 TDP1 (0.42) LMNAMAPTNPSR1ALDH1A1MEN1
SCHEMBL29812171 0.69 PRKCZ (0.34) MAPTPRKCZTRPM8NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1064283-A1 PYRAZOLO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2001-01-03 EP disclosed
WO-1999048892-A1 PYRAZOLO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1999-09-30 WO disclosed