SCHEMBL2659360

SCHEMBL2659360

CC(C)(C)OC(=O)c1cccnc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.60
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
TDP1 Q9NUW8 3/20 0.56
L3MBTL1 Q9Y468 2/20 0.52
CYP1A2 P05177 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
CASP3 P42574 1/20 0.51
SENP8 Q96LD8 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
SENP6 Q9GZR1 1/20 0.51
KMT2A Q03164 5/20 0.49
MEN1 O00255 3/20 0.49
ATR Q13535 1/20 0.49
CYP2D6 P10635 1/20 0.48
PKM P14618 1/20 0.48
AGTR1 P30556 1/20 0.47
HTT P42858 1/20 0.47
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29550920 1.00 POLB (0.60) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL27645361 0.83 POLB (0.46) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL30441012 0.81 KDM4E (0.46) POLBLMNATDP1L3MBTL1ALDH1A1
SCHEMBL163493 0.81 POLB (0.45) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL2633213 0.81 P2RX7 (0.56) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL624343 0.81 LMNA (0.61) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL29412879 0.81 LMNA (0.61) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL9837285 0.81 POLB (0.45) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL8422472 0.80 POLB (0.44) POLBLMNASMN1; SMN2TDP1L3MBTL1
SCHEMBL1292847 0.80 NAPRT (0.56) POLBTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250213547-A1 METHODS OF TREATING NEUROLOGICAL DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2025-07-03 US disclosed
US-12012466-B2 Peptide macrocycles against Acinetobacter baumannii HOFFMANN-LA ROCHE INC. (US) 2024-06-18 US disclosed
CN-117843619-A Modulators of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and methods for preparing the modulators 弗特克斯药品有限公司 2024-04-09 CN disclosed
CN-110267948-B Modulators of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and methods for preparing the modulators 弗特克斯药品有限公司 2023-12-08 CN disclosed
WO-2023175591-A1 METHODS OF TREATING NEUROLOGICAL DISEASES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-09-21 WO disclosed
CN-115872926-A Preparation method of triazole antifungal drug and intermediate thereof 南通诺泰生物医药技术有限公司 2023-03-31 CN disclosed
CN-115772121-A Preparation method of 2-methylamino-3-hydroxymethylpyridine 南通诺泰生物医药技术有限公司 2023-03-10 CN disclosed
US-20220411468-A1 PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII HOFFMANN-LA ROCHE INC. (US) 2022-12-29 US disclosed
US-11447449-B2 Inhibitors of indoleamine 2,3-dioxygenase and methods of their use BRISTOL-MYERS SQUIBB COMPANY (US) 2022-09-20 US disclosed
CN-109803962-B Modulators of cystic fibrosis transmembrane conductance regulator proteins, and pharmaceutical compositions 弗特克斯药品有限公司 2022-04-29 CN disclosed
US-6812238-B1 WATER SOLUBLE FUNGICIDES FOR SYSTEMIC MYCOSES; ORAL AND PARENTERAL ADMINISTRATION BASILEA PHARMACEUTICA AG (CH) 2004-11-02 US disclosed
US-6812238-B1 WATER SOLUBLE FUNGICIDES FOR SYSTEMIC MYCOSES; ORAL AND PARENTERAL ADMINISTRATION BASILEA PHARMACEUTICA AG (CH) 2004-11-02 US disclosed
US-6562844-B2 Attaching an olefin to a solid support; oxidizing the olefin to provide an epoxide functionality; opening the epoxide with an amine to form an amino alcohol; cyclizing the amino alcohol using a phosgene equivalent PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed
US-6531470-B1 Antimicrobial compounds PHARMACIA & UPJOHN COMPANY 2003-03-11 US disclosed
EP-1280795-A2 N-SUBSTITUTED CARBAMOYLOXYALKYL-AZOLIUM DERIVATIVES Basilea Pharmaceutica AG (CH) 2003-02-05 EP disclosed
US-20020183371-A1 Oxazolidinone combinatorial libraries, compositions and methods of preparation GORDEEV MIKHAIL F (US) 2002-12-05 US disclosed
US-6239152-B1 Oxazolidinone combinatorial libraries, compositions and methods of preparation PHARMACIA & UPJOHN COMPANY 2001-05-29 US disclosed
WO-2001032652-A2 N-SUBSTITUTED CARBAMOYLOXYALKYL-AZOLIUM DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2001-05-10 WO disclosed
EP-1049682-A1 OXAZOLIDINONE COMBINATORIAL LIBRARIES, COMPOSITIONS AND METHODS OF PREPARATION Versicor, Inc. (US) 2000-11-08 EP disclosed
WO-1999037630-A1 OXAZOLIDINONE COMBINATORIAL LIBRARIES, COMPOSITIONS AND METHODS OF PREPARATION VERSICOR, INC. (US) 1999-07-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020183371-A1 Oxazolidinone combinatorial libraries, compositions and methods of preparation PAICS, CDK4, OXA1L POLB 307/4885LMNA 1648/4885SMN1; SMN2 154/4885
US-20220411468-A1 PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII VIP, ARG1, CX3CR1 POLB 3834/4885LMNA 3944/4885SMN1; SMN2 4573/4885
US-12012466-B2 Peptide macrocycles against Acinetobacter baumannii VIP, ARG1, CX3CR1 POLB 3834/4885LMNA 3944/4885SMN1; SMN2 4573/4885
US-20250213547-A1 METHODS OF TREATING NEUROLOGICAL DISEASES SMN1; SMN2, PMP22, GBA2 POLB 2602/4885LMNA 2937/4885SMN1; SMN2 1/4885
US-11447449-B2 Inhibitors of indoleamine 2,3-dioxygenase and methods of their use IDO1, IDO2, INMT POLB 1958/4885LMNA 4537/4885SMN1; SMN2 4367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.