SCHEMBL2660397

SCHEMBL2660397

Cc1cc(NS(=O)(=O)c2sccc2C)c2[nH]c(C(=O)NCC(/C=N/O)SCc3ccccc3)cc2c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.31
PYGL P06737 1/20 0.31
LGALS8 O00214 1/20 0.31
LGALS3 P17931 1/20 0.31
CA1 P00915 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659767 0.93 PYGL (0.32) MCL1PYGLLGALS8LGALS3CA1
SCHEMBL2660472 0.89 PLA2G7 (0.31) MCL1
SCHEMBL2659747 0.88 MCL1 (0.31) MCL1PYGLLGALS8LGALS3CA1
SCHEMBL2661002 0.86 LGALS8 (0.32) PYGLLGALS8LGALS3
SCHEMBL2660563 0.86 HDAC3 (0.36)
SCHEMBL2659987 0.82 LGALS8 (0.33) MCL1LGALS8LGALS3
SCHEMBL2660852 0.81 PLA2G7 (0.33) MCL1
SCHEMBL2967882 0.78 TP53 (0.33) PYGL
SCHEMBL2660398 0.78 TP53 (0.33) PYGL
SCHEMBL2660519 0.78 HDAC3 (0.35) LGALS8LGALS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed