SCHEMBL2659987

SCHEMBL2659987

Cc1ccsc1S(=O)(=O)Nc1cc(OC(F)(F)F)cc2cc(C(=O)NCC(C=O)SCc3ccccc3)[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LGALS8 O00214 1/20 0.33
LGALS3 P17931 1/20 0.33
HDAC1 Q13547 2/20 0.32
HDAC3 O15379 1/20 0.32
MCL1 Q07820 9/20 0.32
SLC40A1 Q9NP59 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
HDAC2 Q92769 1/20 0.31
NAMPT P43490 1/20 0.31
KDM4E B2RXH2 3/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
ITGB3 P05106 1/20 0.30
ITGA2B P08514 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2661758 0.90 LGALS8 (0.32) LGALS8LGALS3HDAC1HDAC3MCL1
SCHEMBL2659767 0.89 PYGL (0.32) LGALS8LGALS3MCL1HDAC2KMT2A
SCHEMBL2660563 0.87 HDAC3 (0.36) HDAC1HDAC3
SCHEMBL2659802 0.86 CTSS (0.32) MCL1KDM4E
SCHEMBL2660852 0.83 PLA2G7 (0.33) MCL1KMT2A
SCHEMBL2660397 0.82 MCL1 (0.31) LGALS8LGALS3MCL1
SCHEMBL2659681 0.80 SLC40A1 (0.37) LGALS8LGALS3MCL1SLC40A1KDM4E
SCHEMBL2660539 0.79 MMP13 (0.40) LGALS8LGALS3SLC40A1KDM4EGAA
SCHEMBL2661002 0.79 LGALS8 (0.32) LGALS8LGALS3KDM4EKMT2A
SCHEMBL2659988 0.79 NAMPT (0.34) HDAC1HDAC3HDAC2NAMPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed