SCHEMBL2660508

SCHEMBL2660508

Cc1cccnc1S(=O)(=O)Nc1cc(OCCCS(C)(=O)=O)cc2cc(C(=O)NCC(CN3CCOCC3)SCc3ccccc3)[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.33
ITGB3 P05106 3/20 0.33
ITGA2B P08514 3/20 0.33
MCL1 Q07820 1/20 0.33
MAPT P10636 4/20 0.32
KDM4E B2RXH2 3/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LMNA P02545 3/20 0.32
TP53 P04637 3/20 0.32
THRB P10828 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 3/20 0.31
AVPR1B P47901 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659492 0.93 ITGB3 (0.33) ITGB3ITGA2BMAPTLMNATP53
SCHEMBL2660035 0.93 ITGB3 (0.33) ITGB3ITGA2BMAPTLMNATP53
SCHEMBL2659562 0.93 DRD2 (0.33) ITGB3ITGA2BMAPTLMNATP53
SCHEMBL2668802 0.92 ITGB3 (0.33) SYKITGB3ITGA2BMCL1MAPT
SCHEMBL2662038 0.87 LMNA (0.38) SYKMAPTKDM4ENPSR1LMNA
SCHEMBL2659937 0.87 ITGB3 (0.33) ITGB3ITGA2BMAPTLMNATP53
SCHEMBL2660667 0.86 MAPT (0.35) ITGB3ITGA2BMAPTLMNATP53
SCHEMBL2658758 0.84 MAPT (0.33) ITGB3ITGA2BMCL1MAPTKDM4E
SCHEMBL2668612 0.84 ITGB3 (0.33) ITGB3ITGA2B
SCHEMBL2659399 0.83 SYK (0.32) SYKITGB3ITGA2BMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed