SCHEMBL2668575

SCHEMBL2668575

COC(OC)C(CNC(=O)c1cc2c(C)ccc(NS(=O)(=O)c3cccs3)c2[nH]1)SCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2A1 Q16548 3/20 0.41
MCL1 Q07820 2/20 0.39
BCL2 P10415 1/20 0.37
BID P55957 1/20 0.37
BCL2L1 Q07817 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
BCL2L2 Q92843 1/20 0.37
ALDH1A1 P00352 4/20 0.37
BRD4 O60885 3/20 0.37
FBP1 P09467 1/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
TP53 P04637 2/20 0.36
TNF P01375 1/20 0.35
MAPK1 P28482 1/20 0.35
NOD2 Q9HC29 1/20 0.35
NOD1 Q9Y239 1/20 0.35
USP2 O75604 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2661327 0.90 PLA2G7 (0.31) MEN1KMT2ALMNAPOLB
SCHEMBL2659947 0.88 ALDH1A1 (0.40) BCL2A1MCL1BCL2BIDBCL2L1
SCHEMBL2661328 0.85 TP53 (0.35) ALDH1A1FBP1MAPTMEN1KMT2A
SCHEMBL2660519 0.79 HDAC3 (0.35) MAPTTP53LMNATHRB
SCHEMBL2661002 0.77 LGALS8 (0.32) MAPTMEN1KMT2A
SCHEMBL2660521 0.77 PLCG2 (0.37) ALDH1A1FBP1MAPTMEN1KMT2A
SCHEMBL2661004 0.77 RAB9A (0.34) ALDH1A1MAPTMEN1KMT2ATP53
SCHEMBL2660852 0.77 PLA2G7 (0.33) MCL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL1655516 0.76 BRAF (0.46) BCL2A1MCL1BCL2BIDBCL2L1
SCHEMBL2660809 0.76 PLA2G7 (0.33) MCL1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed