SCHEMBL267933

SCHEMBL267933

COc1ccccc1CCC(C)N

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.61
SLC6A2 P23975 1/20 0.58
SLC6A4 P31645 1/20 0.58
SLC6A3 Q01959 1/20 0.58
AOC3 Q16853 1/20 0.54
IDO1 P14902 2/20 0.52
SIGMAR1 Q99720 1/20 0.50
KMT2A Q03164 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA5A P35218 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
KCNH2 Q12809 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
HRH3 Q9Y5N1 1/20 0.47
ABCB1 P08183 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30520870 1.00 TAAR1 (0.61) TAAR1SLC6A2SLC6A4SLC6A3AOC3
SCHEMBL28089294 0.89 TAAR1 (0.58) TAAR1AOC3IDO1SIGMAR1KMT2A
SCHEMBL7636733 0.85 TAAR1 (0.60) TAAR1AOC3IDO1SIGMAR1CA12
SCHEMBL31147801 0.85 TAAR1 (0.60) TAAR1AOC3IDO1SIGMAR1CA12
SCHEMBL30392457 0.84 CA12 (0.52) TAAR1SLC6A2SLC6A4SLC6A3CA12
SCHEMBL268369 0.84 CA12 (0.52) TAAR1SLC6A2SLC6A4SLC6A3CA12
SCHEMBL23259489 0.81 TAAR1 (0.56) TAAR1AOC3IDO1SIGMAR1CA12
SCHEMBL7535470 0.81 TAAR1 (0.56) TAAR1AOC3IDO1SIGMAR1KCNH2
SCHEMBL14655700 0.81 KMT2A (0.64) TAAR1IDO1KMT2A
SCHEMBL30249073 0.81 KMT2A (0.64) TAAR1IDO1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250186369-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATING, AMELIORATING, AND/OR PRVENTING COCAINE USE DISORDER UNIV DREXEL (US) 2025-06-12 US claimed
US-20240074993-A1 METHODS OF TREATING OR PREVENTING AN ATTENTION DISORDER, COGNITIVE DISORDER, AND/OR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER UNIV DREXEL (US) 2024-03-07 US claimed
WO-2023172497-A2 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATING, AMELIORATING, AND/OR PREVENTING COCAINE USE DISORDER DREXEL UNIVERSITY (US) 2023-09-14 WO claimed
US-20220233475-A1 NOVEL D3 DOPAMINE RECEPTOR AGONISTS TO TREAT DYSKINESIA IN PARKINSON'S DISEASE UNIV DREXEL (US) 2022-07-28 US claimed
US-10695302-B2 Treatments for attention and cognitive disorders, and for dementia associated with a neurodegenerative disorder DREXEL UNIVERSITY (US) 2020-06-30 US claimed
EP-3062791-B1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER UNIV DREXEL (US) 2020-01-08 EP claimed
US-20180092865-A1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER DREXEL UNIVERSITY (US) 2018-04-05 US claimed
US-9861594-B2 Treatments for attention and cognitive disorders, and for dementia associated with a neurodegenerative disorder DREXEL UNIVERSITY (US) 2018-01-09 US claimed
US-9675565-B2 D3 dopamine receptor agonists to treat dyskinesia in parkinson's disease DREXEL UNIVERSITY (US) 2017-06-13 US claimed
US-20160256417-A1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER DREXEL UNIVERSITY (US) 2016-09-08 US claimed
EP-3062791-A1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER Drexel University (US) 2016-09-07 EP claimed
US-9289400-B2 D3 dopamine receptor agonists to treat dyskinesia in parkinson's disease DREXEL UNIVERSITY (US) 2016-03-22 US claimed
WO-2015066019-A1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER DREXEL UNIVERSITY (US) 2015-05-07 WO claimed
US-20140228355-A1 Novel D3 Dopamine Receptor Agonists to Treat Dyskinesia in Parkinson's Disease UNIVERSITY OF MEDICINE AND DENTISTRY NEW JERSEY MEDICAL SCHOOL (US) 2014-08-14 US claimed
US-20140228380-A1 Novel D3 Dopamine Receptor Agonists to Treat Dyskinesia in Parkinson's Disease UNIVERSITY OF MEDICINE AND DENTISTRY NEW JERSEY MEDICAL SCHOOL (US) 2014-08-14 US claimed
EP-2603215-A2 NOVEL D3 DOPAMINE RECEPTOR AGONISTS TO TREAT DYSKINESIA IN PARKINSON'S DISEASE Philadelphia Health and Education Corporation (US) 2013-06-19 EP claimed
WO-2012021629-A2 NOVEL D3 DOPAMINE RECEPTOR AGONISTS TO TREAT DYSKINESIA IN PARKINSON'S DISEASE PHILADELPHIA HEALTH & EDUCATION CORPORATION (US) 2012-02-16 WO claimed
US-20250186369-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATING, AMELIORATING, AND/OR PRVENTING COCAINE USE DISORDER UNIV DREXEL (US) 2025-06-12 US disclosed
US-4563458-A CIRCULATORY SYSTEM DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1986-01-07 US disclosed
EP-0114374-A1 Substituted 4-aminomethylene chromans or chromenes, process for their preparation and their use in medicines BAYER AG (DE) 1984-08-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10695302-B2 Treatments for attention and cognitive disorders, and for dementia associated with a neurodegenerative disorder CHAT, ACHE, SLC18A3 TAAR1 533/4885SLC6A2 10/4885SLC6A4 23/4885
US-20240074993-A1 METHODS OF TREATING OR PREVENTING AN ATTENTION DISORDER, COGNITIVE DISORDER, AND/OR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER CHAT, COMT, SLC6A2 TAAR1 590/4885SLC6A2 3/4885SLC6A4 15/4885
US-20220233475-A1 NOVEL D3 DOPAMINE RECEPTOR AGONISTS TO TREAT DYSKINESIA IN PARKINSON'S DISEASE DRD3, PARK7, SLC6A3 TAAR1 206/4885SLC6A2 128/4885SLC6A4 235/4885
US-20140228380-A1 Novel D3 Dopamine Receptor Agonists to Treat Dyskinesia in Parkinson's Disease DRD3, PARK7, SLC6A3 TAAR1 206/4885SLC6A2 128/4885SLC6A4 235/4885
US-20180092865-A1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER CHAT, BDNF, SLC18A3 TAAR1 355/4885SLC6A2 13/4885SLC6A4 26/4885
US-20160256417-A1 NOVEL TREATMENTS FOR ATTENTION AND COGNITIVE DISORDERS, AND FOR DEMENTIA ASSOCIATED WITH A NEURODEGENERATIVE DISORDER CHAT, BDNF, SLC18A3 TAAR1 355/4885SLC6A2 13/4885SLC6A4 26/4885
US-20250186369-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATING, AMELIORATING, AND/OR PRVENTING COCAINE USE DISORDER CES2, CHAT, SLC18A2 TAAR1 110/4885SLC6A2 7/4885SLC6A4 33/4885
US-20140228355-A1 Novel D3 Dopamine Receptor Agonists to Treat Dyskinesia in Parkinson's Disease DRD3, PARK7, SLC6A3 TAAR1 206/4885SLC6A2 128/4885SLC6A4 235/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.