SCHEMBL268678

SCHEMBL268678

CON(C)C(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
CA12 O43570 4/20 0.39
CA2 P00918 4/20 0.39
CA14 Q9ULX7 2/20 0.39
JAK3 P52333 1/20 0.37
BTK Q06187 1/20 0.37
PRMT3 O60678 1/20 0.36
CA1 P00915 4/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
EPHX1 P07099 1/20 0.36
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18176811 0.84 TDP1 (0.43) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL1328516 0.83 TDP1 (0.46) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL2795678 0.83 TDP1 (0.47) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL3683152 0.81 TDP1 (0.44) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL4235641 0.80 TDP1 (0.38) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL895070 0.80 TDP1 (0.53) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL500234 0.79 TDP1 (0.55) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL21887790 0.79 MEN1 (0.43) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL31270901 0.78 CA12 (0.43) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL20524433 0.78 KMT2A (0.38) MEN1KMT2AGAAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 450 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260124204-A1 METALLOENZYME INHIBITOR COMPOUNDS EIKONIZO THERAPEUTICS, INC. (US) 2026-05-07 US disclosed
US-12617762-B2 Carboxy derivatives with antiinflamatory properties SITRYX THERAPEUTICS LIMITED (GB) 2026-05-05 US disclosed
US-20260092063-A1 FUSED BICYCLIC RAF INHIBITORS AND METHODS FOR USE THEREOF JAZZ PHARMACEUTICALS IRELAND LTD (IE) 2026-04-02 US disclosed
EP-4081511-B3 CARBOXY DERIVATIVES WITH ANTIINFLAMMATORY PROPERTIES SITRYX THERAPEUTICS LTD (GB) 2026-03-04 EP disclosed
EP-4655302-A1 TYRO3 SELECTIVE INHIBITORS AND USES THEREOF The University of North Carolina at Chapel Hill (US) 2025-12-03 EP disclosed
WO-2025244832-A1 NOVEL AMINOGUANIDINE DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF KONG'S PHARMACEUTICAL CO. (US) 2025-11-27 WO disclosed
US-12398120-B2 Substituted hydantoinamides as ADAMTS7 antagonists BAYER AKTIENGESELLSCHAFT (DE) 2025-08-26 US disclosed
US-12370194-B2 Metalloenzyme inhibitor compounds EIKONIZO THERAPEUTICS, INC. (US) 2025-07-29 US disclosed
EP-4562001-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS Nura Bio, Inc. (US) 2025-06-04 EP disclosed
US-12304912-B2 Fused bicyclic RAF inhibitors and methods for use thereof JAZZ PHARMACEUTICALS IRELAND LIMITED (IE) 2025-05-20 US disclosed
CN-1440385-A Pyrrole derivatives for the treatment of AIDS HOFFMANN LA ROCHE (CH) 2003-09-03 CN disclosed
WO-2003053971-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2003-07-03 WO disclosed
EP-1301481-A1 PYRROLE DERIVATIVES FOR TREATING AIDS F. HOFFMANN-LA ROCHE AG (CH) 2003-04-16 EP disclosed
US-6534530-B1 Administering (benzo)thiazole peptidomimetic as viricide; protease inhibitors AGOURON PHARMACEUTICALS, INC. 2003-03-18 US disclosed
WO-2003013526-A1 ANTICOAGULANT COMPOUNDS MERCK & CO. INC. (US) 2003-02-20 WO disclosed
US-20020147229-A1 Pharmaceuticals PFIZER INC. 2002-10-10 US disclosed
EP-1242426-A1 GAMMA-HYDROXY-2-(FLUOROALKYLAMINOCARBONYL)-1-PIPERAZINEPENTANAMIDES AS HIV PROTEASE INHIBITORS Merck & Co., Inc. (US) 2002-09-25 EP disclosed
US-20020032221-A1 Pyrrole derivatives ROCHE PRODUCTS LIMITED (GB) 2002-03-14 US disclosed
WO-2002002524-A1 PYRROLE DERIVATIVES FOR TREATING AIDS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-10 WO disclosed
WO-2001038332-A1 GAMMA-HYDROXY-2-(FLUOROALKYLAMINOCARBONYL)-1-PIPERAZINEPENTANAMIDES AS HIV PROTEASE INHIBITORS MERCK & CO., INC. (US) 2001-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12304912-B2 Fused bicyclic RAF inhibitors and methods for use thereof BRAF, RAF1, NRAS TDP1 1065/4885MAOA 1519/4885MAOB 1093/4885
US-12398120-B2 Substituted hydantoinamides as ADAMTS7 antagonists ADAMTS7, MMP7, ADAM17 TDP1 388/4885MAOA 1338/4885MAOB 1041/4885
US-20020032221-A1 Pyrrole derivatives PYCR1, SARS1, MAVS TDP1 990/4885MAOA 3894/4885MAOB 3193/4885
US-20260124204-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC3, HDAC1 TDP1 2647/4885MAOA 155/4885MAOB 106/4885
US-12617762-B2 Carboxy derivatives with antiinflamatory properties CCR1, CBR1, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 TDP1 1053/4885MAOA 2014/4885MAOB 2819/4885
US-20260092063-A1 FUSED BICYCLIC RAF INHIBITORS AND METHODS FOR USE THEREOF BRAF, NRAS, RAF1 TDP1 2146/4885MAOA 1727/4885MAOB 1184/4885
US-20020147229-A1 Pharmaceuticals BDKRB1, TFPI, BDKRB2 TDP1 281/4885MAOA 288/4885MAOB 203/4885
US-12370194-B2 Metalloenzyme inhibitor compounds HDAC6, HDAC1, HDAC2 TDP1 1641/4885MAOA 545/4885MAOB 828/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.