SCHEMBL2724813

SCHEMBL2724813

O=C(O)c1ncc(-c2cccnc2)o1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 1/20 0.55
NPC1 O15118 1/20 0.55
HPGD P15428 1/20 0.55
RAB9A P51151 1/20 0.55
HSD17B10 Q99714 1/20 0.55
FAAH O00519 3/20 0.54
MKNK1 Q9BUB5 2/20 0.50
MKNK2 Q9HBH9 2/20 0.50
KMO O15229 2/20 0.48
CYP3A4 P08684 3/20 0.46
CYP2A6 P11509 3/20 0.46
CYP2E1 P05181 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2B6 P20813 2/20 0.46
CYP2C19 P33261 2/20 0.46
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
TUBB4A P04350 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5105714 0.98 ALDH1A1 (0.54) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL27768674 0.89 FAAH (0.55) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL892926 0.84 TUBB4A (0.59) ALDH1A1KDM4ENPC1HPGDRAB9A
Lithium Ion SCHEMBL5105709 0.84 FAAH (0.52) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL4790263 0.83 TUBB4A (0.57) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL14192604 0.81 FAAH (0.50) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL5109428 0.80 FAAH (0.49) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL5111369 0.79 FAAH (0.56) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL2779211 0.79 FAAH (0.71) FAAHCES1
SCHEMBL2724814 0.77 ALDH1A1 (0.51) ALDH1A1KDM4ENPC1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630133-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-08-28 EP disclosed
WO-2012052412-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-04-26 WO disclosed
US-20080103170-A1 Nicotinic Acetylcholine Receptor Ligands ASTRAZENECA AB (SE) 2008-05-01 US disclosed
US-20070249588-A1 Nicotinic Acetylcholine Receptor Ligands ASTRAZENECA AB (SE) 2007-10-25 US disclosed
EP-1699801-A1 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AstraZeneca AB (SE) 2006-09-13 EP disclosed
WO-2005061510-A1 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2005-07-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080103170-A1 Nicotinic Acetylcholine Receptor Ligands CHRNG, CHRNE, CHRNA1 ALDH1A1 1028/4885KDM4E 2378/4885NPC1 1205/4885
US-20070249588-A1 Nicotinic Acetylcholine Receptor Ligands CHRNA1, CHRNB1, CHRNA2 ALDH1A1 500/4885KDM4E 3396/4885NPC1 1175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.