SCHEMBL27263418

SCHEMBL27263418

Cn1ncc(N2CCN(CCNc3ccccc3F)CC2)c(Cl)c1=O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.46
BRD9 Q9H8M2 2/20 0.46
PKM P14618 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 1/20 0.45
HTR1A P08908 5/20 0.45
ADRA1D P25100 5/20 0.45
ADRA1A P35348 5/20 0.45
ADRA1B P35368 5/20 0.45
KAT2B Q92831 3/20 0.45
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
HRH1 P35367 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TRPC5 Q9UL62 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27263186 0.88 ALDH1A1 (0.47) BRD4BRD9PKMALDH1A1NPC1
SCHEMBL9527005 0.88 ADRA1A (0.52) BRD4BRD9HTR1AADRA1DADRA1A
SCHEMBL27263520 0.86 KAT2B (0.57) BRD4BRD9PKMALDH1A1NPC1
SCHEMBL27263994 0.86 HTR1A (0.57) HTR1AADRA1DADRA1AADRA1B
SCHEMBL27263977 0.85 BRD4 (0.41) BRD4BRD9ALDH1A1HTR1AADRA1D
SCHEMBL27264116 0.84 HTR1A (0.48) HTR1AADRA1DADRA1AADRA1B
SCHEMBL27264164 0.84 BPTF (0.52) BRD4PKMALDH1A1NPC1KAT2B
SCHEMBL27263628 0.84 ADRA1A (0.47) BRD4BRD9ALDH1A1HTR1AADRA1D
SCHEMBL27263416 0.82 HTR1A (0.47) BRD4BRD9HTR1AADRA1DADRA1A
SCHEMBL9528374 0.82 DRD2 (0.58) BRD4BRD9HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1022565-C Process for preparing piperazinylalkyl-3(2H)-pyridazinones CL PHARMA (AT) 1993-10-27 CN disclosed
CN-1043129-A New piperazinyl alkyl-3 (2H)-pyridazinone, its preparation method and as the application of hypotensive agent CL PHARMA (AT) 1990-06-20 CN disclosed