SCHEMBL2726428

SCHEMBL2726428

Cc1csc([C@H]2CCCN2C(=O)c2cc(C(=O)NN)n(C)c(=O)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAA50 Q9GZZ1 5/20 0.39
POLB P06746 1/20 0.37
TRPV1 Q8NER1 3/20 0.37
BAZ2A Q9UIF9 1/20 0.36
HSD11B1 P28845 2/20 0.36
TSHR P16473 1/20 0.36
KDM4E B2RXH2 2/20 0.35
USP2 O75604 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
CPT2 P23786 1/20 0.33
CPT1A P50416 1/20 0.33
CPT1B Q92523 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2726484 0.88 NAA50 (0.39) NAA50POLBTRPV1BAZ2AHSD11B1
SCHEMBL2725263 0.85 NAA50 (0.42) NAA50POLBTRPV1BAZ2AHSD11B1
SCHEMBL6467555 0.84 TRPV1 (0.41) NAA50POLBTRPV1BAZ2ATSHR
SCHEMBL10289968 0.82 TRPV1 (0.39) POLBTRPV1BAZ2ATSHRKDM4E
SCHEMBL6467840 0.82 AADAT (0.39) NAA50POLBTRPV1
SCHEMBL10290632 0.81 TRPV1 (0.39) NAA50POLBTRPV1BAZ2ATSHR
SCHEMBL2726629 0.81 TRPV1 (0.39) NAA50POLBTRPV1BAZ2ATSHR
SCHEMBL6466071 0.81 POLB (0.38) NAA50POLBTRPV1BAZ2ATSHR
SCHEMBL2727029 0.81 HSD11B1 (0.37) NAA50POLBTRPV1BAZ2AHSD11B1
SCHEMBL2727621 0.80 NAA50 (0.38) NAA50POLBTRPV1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed