SCHEMBL2729239

SCHEMBL2729239

NC(=O)c1cnn(-c2ccc(N)cc2F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.43
BTK Q06187 2/20 0.40
MAP4K4 O95819 1/20 0.37
MAPT P10636 2/20 0.36
GFER P55789 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
THRB P10828 1/20 0.36
ALOX15 P16050 1/20 0.36
YWHAG P61981 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SYK P43405 1/20 0.36
HPGDS O60760 1/20 0.36
ALKBH2 Q6NS38 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10139201 0.84 CYP1A2 (0.52) ACKR3MAPTKDM4EHSD17B10CYP1A2
SCHEMBL3758177 0.81 CYP1A2 (0.47) ACKR3MAPTMEN1ALOX15KMT2A
SCHEMBL13054790 0.81 ACKR3 (0.39) ACKR3MAPTGFERCYP1A2CYP3A4
SCHEMBL27835961 0.81 ALKBH2 (0.45) BTKMAP4K4MAPTHPGDSALKBH2
SCHEMBL14320344 0.76 TDO2 (0.49) MAPTGFERKDM4EMEN1THRB
SCHEMBL10139147 0.75 MAP4K4 (0.56) BTKMAP4K4MAPTKDM4EMEN1
SCHEMBL4647029 0.74 ALKBH1 (0.56) ACKR3HPGDSALKBH2EGLN1NPC1
SCHEMBL30132085 0.74 HPGDS (0.51) BTKMAP4K4MAPTMEN1KMT2A
SCHEMBL4481678 0.74 HPGDS (0.51) BTKMAP4K4MAPTMEN1KMT2A
SCHEMBL30529091 0.74 ALKBH1 (0.56) ACKR3HPGDSALKBH2EGLN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059932-A1 2, 4 -DIAMINOPYRIMIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2012-05-10 WO disclosed
WO-2012059932-A1 2, 4 -DIAMINOPYRIMIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2012-05-10 WO disclosed