SCHEMBL27362044

SCHEMBL27362044

CC(C)c1cc(CC(C)c2cncc(C(=O)O)n2)cc(C(=O)O)n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
KDM4E B2RXH2 1/20 0.33
HMGCR P04035 1/20 0.32
PTGER1 P34995 1/20 0.31
COPS5 Q92905 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
HIF1A Q16665 1/20 0.31
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20967854 0.79 HMGCR (0.35) HMGCRTSHRESR1ESR2
SCHEMBL1760148 0.79 KDM4E (0.41) HCAR3HCAR2KDM4EALOX15TSHR
SCHEMBL17465991 0.68 NOS3 (0.50) HCAR3HCAR2KDM4EPTGER1ALOX15
SCHEMBL3087546 0.66 HCAR3 (0.44) HCAR3HCAR2KDM4EALOX15TSHR
SCHEMBL16369768 0.66 HCAR2 (0.41) HCAR2KDM4EALOX15TSHRHIF1A
SCHEMBL19151634 0.65 ADORA3 (0.42) TSHR
SCHEMBL31636273 0.65 ADORA3 (0.42) TSHR
SCHEMBL24993310 0.64 P2RX7 (0.41) KDM4E
SCHEMBL1425522 0.64 ALDH1A1 (0.40) KDM4EALOX15TSHRHIF1AESR1
SCHEMBL69399 0.64 KDM4E (0.55) HCAR2KDM4EALOX15TSHRHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023235753-A2 ALDH2 INHIBITORS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-12-07 WO disclosed