SCHEMBL27363608

SCHEMBL27363608

CCCCCON(CC(=O)O)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.43
CYP3A4 P08684 3/20 0.43
MAPK1 P28482 3/20 0.43
TP53 P04637 1/20 0.43
PLA2G2A P14555 1/20 0.43
BLM P54132 1/20 0.43
CYSLTR2 Q9NS75 2/20 0.42
CYSLTR1 Q9Y271 2/20 0.42
LTA4H P09960 1/20 0.42
LMNA P02545 4/20 0.42
ALDH1A1 P00352 2/20 0.42
CETP P11597 3/20 0.41
MEN1 O00255 1/20 0.41
NR1I2 O75469 1/20 0.41
CHRM2 P08172 1/20 0.41
ADRA2A P08913 1/20 0.41
MAPT P10636 1/20 0.41
OPRK1 P41145 1/20 0.41
HTR2B P41595 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10770087 0.86 LTA4H (0.44) TSHRCYP3A4MAPK1TP53LTA4H
SCHEMBL10171416 0.79 PLA2G2A (0.49) TSHRPLA2G2ABLMALDH1A1MEN1
SCHEMBL2945289 0.79 TSHR (0.47) TSHRCYP3A4MAPK1TP53LMNA
SCHEMBL10351423 0.78 TSHR (0.48) TSHRCYP3A4MAPK1TP53LTA4H
SCHEMBL345325 0.76 PLA2G2A (0.46) TSHRPLA2G2ABLMALDH1A1MEN1
SCHEMBL28253232 0.76 NPC1 (0.46) TSHRMAPK1LMNAALDH1A1MEN1
SCHEMBL10777388 0.75 ALDH1A1 (0.43) TSHRLMNAALDH1A1MEN1MAPT
SCHEMBL9417494 0.75 PLA2G2A (0.50) TSHRCYP3A4MAPK1TP53PLA2G2A
SCHEMBL9417618 0.75 PLA2G2A (0.50) TSHRCYP3A4MAPK1TP53PLA2G2A
SCHEMBL2368553 0.74 TSHR (0.45) TSHRCYP3A4MAPK1TP53LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1078968-A 2-Piperazinone compounds and their preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1993-12-01 CN disclosed
CN-1069730-A 2-Piperazinone compounds and their preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1993-03-10 CN disclosed