SCHEMBL27368430

SCHEMBL27368430

CCc1cc(NCc2ccc(C#N)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 4/20 0.42
EPHX2 P34913 1/20 0.37
CYP19A1 P11511 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
HIF1A Q16665 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
AKR1B1 P15121 1/20 0.36
CISD1 Q9NZ45 2/20 0.35
CYP2A6 P11509 1/20 0.35
KLKB1 P03952 1/20 0.35
KLK1 P06870 1/20 0.35
RORC P51449 1/20 0.35
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
MAPK10 P53779 1/20 0.34
PDE5A O76074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27348369 0.89 VNN1 (0.41) VNN1MAPK8
SCHEMBL27348370 0.88 VNN1 (0.43) VNN1EPHX2CYP19A1LOXL2HIF1A
SCHEMBL8635360 0.84 TBXA2R (0.41)
SCHEMBL27369277 0.82 SCN1A (0.39)
SCHEMBL8632351 0.77 PDE4B (0.41)
SCHEMBL27352876 0.77 VNN1 (0.42) VNN1
SCHEMBL8633057 0.75 L3MBTL1 (0.41)
SCHEMBL8634221 0.75 SIRT2 (0.34) RORC
SCHEMBL27347115 0.71 SCN1A (0.39) KLKB1
SCHEMBL8538752 0.71 SLC9A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed