Fatostatin

Fatostatin

SCHEMBL2742732

CCCc1cc(-c2nc(-c3ccc(C)cc3)cs2)ccn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SREBF2 Q12772 17/20 1.00
MAPT P10636 3/20 0.97
ATM Q13315 3/20 0.97
L3MBTL1 Q9Y468 2/20 0.97
ALDH1A1 P00352 1/20 0.97
SREBF1 P36956 2/20 0.81
KDM4E B2RXH2 2/20 0.77
LMNA P02545 2/20 0.77
RECQL P46063 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fatostatin SCHEMBL29458338 1.00 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
Fatostatin SCHEMBL25327929 0.99 MAPT (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL19758233 0.95 SREBF2 (0.90) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4279559 0.89 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4293604 0.88 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4290927 0.88 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4285116 0.88 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4286504 0.88 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4292296 0.88 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1
SCHEMBL4283881 0.88 SREBF2 (1.00) SREBF2MAPTATML3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 136 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230414626-A1 INDUCTION OF FERROPTOSIS FOR CANCER THERAPY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-12-28 US claimed
US-11504390-B2 Treatment of increased lipid levels with sterol regulatory element binding transcription factor 1 (SREBF1) inhibitors REGENERON PHARMACEUTICALS, INC. (US) 2022-11-22 US claimed
WO-2022120197-A1 COMBINATIONS OF EPIDERMAL GROWTH FACTOR RECEPTOR INHIBITORS AND STEROL REGULATORY ELEMENT-BINDING PROTEIN INHIBITORS FOR USES IN CANCER THERAPIES EMORY UNIVERSITY (US) 2022-06-09 WO claimed
WO-2022093770-A1 COMBINATION THERAPY WITH PI3K-AKT-MTOR INHIBITORS AND FERROPTOSIS INDUCING AGENTS TO TREAT CANCER MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-05-05 WO claimed
WO-2022082078-A1 INDUCTION OF FERROPTOSIS FOR CANCER THERAPY MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-04-21 WO claimed
US-20130012538-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2013-01-10 US claimed
US-20130005768-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2013-01-03 US claimed
US-8207196-B2 Compositions and methods for the treatment of metabolic disorders BAYLOR COLLEGE OF MEDICINE (US) 2012-06-26 US claimed
EP-2120580-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS Baylor College Of Medicine (US) 2009-11-25 EP claimed
US-20090131475-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2009-05-21 US claimed
WO-2008097835-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2008-08-14 WO claimed
US-20250297321-A1 METHOD FOR DETECTING METABOLIC REPROGRAMING OF CANCER TOWARDS FATTY ACIDS METABOLISM INST NAT SANTE RECH MED (FR) 2025-09-25 US disclosed
US-12048694-B2 Coordinated metabolic reprogramming in response to productive viral infections ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2024-07-30 US disclosed
US-20230414626-A1 INDUCTION OF FERROPTOSIS FOR CANCER THERAPY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-12-28 US disclosed
US-20230263821-A1 Treatment Of Increased Lipid Levels With Sterol Regulatory Element Binding Transcription Factor 1 (SREBF1) Inhibitors UNIVERSITY OF MARYLAND, BALTIMORE 2023-08-24 US disclosed
WO-2010092153-A1 NEW SUBSTITUTED TETRAHYDRONAPTHALENES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS DRUGS SANOFI-AVENTIS (FR) 2010-08-19 WO disclosed
EP-2120580-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS Baylor College Of Medicine (US) 2009-11-25 EP disclosed
US-20090131475-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2009-05-21 US disclosed
US-20090131475-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2009-05-21 US disclosed
WO-2008097835-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS BAYLOR COLLEGE OF MEDICINE (US) 2008-08-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12048694-B2 Coordinated metabolic reprogramming in response to productive viral infections MAVS, ATF4, PC SREBF2 28/4885MAPT 2780/4885ATM 1642/4885
US-20130012538-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS FABP4, LIPC, FABP1 SREBF2 31/4885MAPT 3510/4885ATM 1753/4885
US-20130005768-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS FABP4, LIPC, FABP1 SREBF2 31/4885MAPT 3510/4885ATM 1753/4885
US-20090131475-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF METABOLIC DISORDERS FABP4, LIPC, FABP1 SREBF2 32/4885MAPT 3438/4885ATM 1694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.