SCHEMBL2743793

SCHEMBL2743793

COc1cc(CO)c(-c2cc3c(cc2CO)OCO3)c(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
GSK3B P49841 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
ATR Q13535 1/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
NQO1 P15559 2/20 0.41
OPRK1 P41145 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31134196 0.84 CYP3A4 (0.42) CYP3A4GSK3BKMT2AMEN1ATR
SCHEMBL31134164 0.84 LMNA (0.55) CYP3A4GSK3BKMT2AMEN1ATR
SCHEMBL5534604 0.78 PDE4A (0.52) CYP3A4
SCHEMBL2743785 0.74 PDE5A (0.49)
SCHEMBL28312125 0.70 PDE4A (0.52) CYP3A4
SCHEMBL7437553 0.70 GSK3B (0.54) GSK3BKMT2AMEN1ATRPOLB
SCHEMBL2743668 0.70 GSK3B (0.51) GSK3BKMT2AMEN1ATRPOLB
SCHEMBL11928777 0.70 PDE4A (0.44) CYP3A4
SCHEMBL2743661 0.69 LMNA (0.60) GSK3BKMT2AMEN1ATRPOLB
SCHEMBL25371015 0.69 CYP3A4 (0.67) CYP3A4POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178578-B2 Chemical compounds THE UNIVERSITY OF MANCHESTER (GB) 2012-05-15 US disclosed
US-20100016261-A1 CHEMICAL COMPOUNDS THE UNIVERSITY OF MANCHESTER (GB) 2010-01-21 US disclosed
EP-2101755-A2 POLYALKYLOXYDIBENZ (C,E) OXEPINE DERIVATIVES AS MEDICAMENTS The University of Manchester (GB) 2009-09-23 EP disclosed
WO-2008075048-A2 POLYALKYLOXYDIBENZ ( C, E) OXEPINE DERIVATIVES AS MEDICAMENTS THE UNIVERSITY OF MANCHESTER (GB) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016261-A1 CHEMICAL COMPOUNDS CYP11B2, MPO, PIGO CYP3A4 138/4885GSK3B 2541/4885KMT2A 3940/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.