SCHEMBL27460897

SCHEMBL27460897

COc1ccccc1-c1csc(OC(C)=O)c1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.39
ALDH1A1 P00352 5/20 0.39
HSD17B10 Q99714 4/20 0.39
HPGD P15428 4/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CYP1A2 P05177 2/20 0.39
TP53 P04637 1/20 0.39
AHR P35869 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ATP4A P20648 2/20 0.39
ATP4B P51164 2/20 0.39
IKBKB O14920 1/20 0.39
FPR1 P21462 2/20 0.38
APP P05067 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
PTK2 Q05397 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27460074 0.82 ALDH1A1 (0.38) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL6998322 0.77 ALDH1A1 (0.46) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL16236644 0.77 KDM4E (0.53) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL8187620 0.76 KDM4E (0.51) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL27729535 0.71 PRKCZ (0.54) KDM4EALDH1A1HSD17B10HPGDIKBKB
SCHEMBL7033578 0.70 ACHE (0.53) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL8676653 0.69 PTGS2 (0.61) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL27374876 0.69 LMNA (0.35) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL4083577 0.69 CA12 (0.50) KDM4EALDH1A1HSD17B10HPGDCYP1A2
SCHEMBL27866713 0.69 GSK3B (0.32) LMNAPRKCZ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1122669-C Novel 8H-thiophene [2,3-b] pyrrolinezine-8-on compound, its preparing method and their medicinal compounds containing them ADIR (FR) 2003-10-01 CN disclosed