SCHEMBL27484813

SCHEMBL27484813

NN=CNc1cccc(C(=O)NCC(=O)NCC(C(=O)O)c2cc(Br)cc(Cl)c2O)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 18/20 0.47
ITGAV P06756 18/20 0.47
ITGB6 P18564 14/20 0.47
ITGB1 P05556 1/20 0.41
ITGA5 P08648 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27503085 0.88 ITGB3 (0.47) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL27555002 0.87 HTT (0.43) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL6777304 0.85 ITGB3 (0.64) ITGB3ITGAVITGB6
SCHEMBL27522236 0.84 ITGB1 (0.41) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7340247 0.82 LMNA (0.43) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL27501985 0.81 ITGB1 (0.44) ITGB3ITGAVITGB1ITGA5MEN1
Propionic Acid SCHEMBL7337742 0.80 LMNA (0.42) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL27484439 0.79 ITGB1 (0.39) ITGB3ITGAVITGB1ITGA5KDM4E
SCHEMBL244092 0.79 ITGB3 (0.68) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7340807 0.78 ITGB3 (0.63) ITGB3ITGAVITGB6ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN claimed