SCHEMBL27504682

SCHEMBL27504682

COC(=O)C(N)c1ccnc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41
PTPN1 P18031 1/20 0.40
PTPN11 Q06124 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
TACR3 P29371 5/20 0.39
HTT P42858 1/20 0.39
HTR2C P28335 3/20 0.39
HTR2B P41595 3/20 0.39
TACR2 P21452 3/20 0.38
TSHR P16473 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28069309 0.81 NCF1 (0.46) NCF1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL13656748 0.77 KMT2A (0.41) ALDH1A1KMT2AMAPT
SCHEMBL6495560 0.77 LOXL2 (0.47) NCF1ALDH1A1CYP1A2PTPN1PTPN11
Hydrochloric Acid SCHEMBL6495563 0.76 LOXL2 (0.46) NCF1ALDH1A1CYP1A2PTPN1PTPN11
SCHEMBL27487557 0.76 MEN1 (0.43) ALDH1A1CYP1A2CYP2C9HIF1AMEN1
Hydrochloric Acid SCHEMBL6495555 0.76 LOXL2 (0.46) NCF1ALDH1A1CYP1A2PTPN1PTPN11
SCHEMBL283103 0.75 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19MEN1
SCHEMBL6302737 0.75 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19MEN1
SCHEMBL9664845 0.75 KMT2A (0.50) ALDH1A1CYP1A2CYP3A4CYP2D6HSD17B10
SCHEMBL264120 0.74 NCF1 (0.52) NCF1ALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1213040-C Serine protease inhibitors LILLY CO ELI (US) 2005-08-03 CN disclosed
CN-1438999-A Serine protease inhibitors LILLY CO ELI (US) 2003-08-27 CN disclosed