Mofebutazone

Mofebutazone

SCHEMBL27513530

CCCCC1C(=O)N(c2ccccc2)N=C1O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
CYP3A4 P08684 2/20 0.57
RAB9A P51151 2/20 0.57
LMNA P02545 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
MAPK1 P28482 1/20 0.57
CYP2C19 P33261 1/20 0.57
TP53 P04637 1/20 0.57
MAPT P10636 1/20 0.57
HPGD P15428 1/20 0.57
PTGS1 P23219 1/20 0.57
NAPRT Q6XQN6 1/20 0.57
CES2 O00748 11/20 0.52
LOX P28300 1/20 0.44
LOXL3 P58215 1/20 0.44
LOXL4 Q96JB6 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
SHMT2 P34897 1/20 0.42
GFER P55789 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylbutazone SCHEMBL28843709 0.94 ALDH1A1 (0.68) ALDH1A1CYP3A4RAB9ALMNACYP1A2
Oxyphenbutazone Anhydrous SCHEMBL28086649 0.89 LMNA (0.77) ALDH1A1CYP3A4RAB9ALMNACYP1A2
SCHEMBL5279293 0.84 CES2 (0.65) ALDH1A1CYP3A4RAB9ALMNACYP1A2
SCHEMBL6700291 0.80 CES2 (0.63) ALDH1A1CYP3A4RAB9ALMNACYP1A2
SCHEMBL9380107 0.76 CES2 (0.46) ALDH1A1CYP3A4RAB9ALMNACYP1A2
SCHEMBL9382481 0.75 CES2 (0.60) MAPTCES2
Phenylbutazone SCHEMBL8005041 0.73 RAB9A (0.82) ALDH1A1CYP3A4RAB9ALMNACYP1A2
Phenylbutazone SCHEMBL3632 0.73 RAB9A (0.82) ALDH1A1CYP3A4RAB9ALMNACYP1A2
Oxyphenbutazone Anhydrous SCHEMBL25857 0.72 LMNA (1.00) ALDH1A1CYP3A4RAB9ALMNACYP1A2
Oxyphenbutazone Anhydrous SCHEMBL5316370 0.72 LMNA (1.00) ALDH1A1CYP3A4RAB9ALMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102143961-B Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activity NEURAXON INC 2014-11-05 CN claimed
CN-102143961-A Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activity NEURAXON INC 2011-08-03 CN claimed
CN-111479575-B Compositions comprising a chemotherapeutic agent and a checkpoint inhibitor and methods of use 北卡罗莱纳州立大学 2024-03-22 CN disclosed
CN-116891540-A Alginic acid derivatives with non-steroidal anti-inflammatory compounds attached thereto 持田制药株式会社 2023-10-17 CN disclosed
CN-116059347-A Treatment and prevention of cancer using HER3 antigen binding molecules 蜂鸟生物科技私人有限公司 2023-05-05 CN disclosed
CN-114945363-A Polyphosphazene drug carriers 昂塞莱克斯制药公司 2022-08-26 CN disclosed
CN-102292449-B Prevent or treat thrombotic IL-6 antagonist ALDER BIOPHARMACEUTICALS, INC. (US) 2016-03-30 CN disclosed
CN-102143961-B Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activity NEURAXON INC 2014-11-05 CN disclosed
CN-101316853-B Benzothiazole and thiazolopyridine as SIRTUIN modulators SIRTRIS PHARMACEUTICALS INC 2014-09-24 CN disclosed
CN-103145738-A Imidazo [2,1-b] thiayole derivatives as SIRTUIN modulating compounds SIRTRIS PHARMACEUTICALS INC 2013-06-12 CN disclosed
CN-102292449-A Antagonists of IL-6 to prevent or treat thrombosis 2011-12-21 CN disclosed
CN-101277963-A Benzimidazole derivatives as SIRTUIN modulators SIRTIS PHARMACEUTICALS INC (US) 2008-10-01 CN disclosed
CN-1898198-A Alpha-hydroxy amides as bradykinin antagonists or inverse agonists MERCK & CO INC (US) 2007-01-17 CN disclosed
CN-1871215-A Cyclic derivatives as modulators of chemokine receptor activity BRISTOL MYERS SQUIBB CO (US) 2006-11-29 CN disclosed
CN-1835944-A Quinolyl amide derivatives as CCR-5 antagonists SCHERING AG (DE) 2006-09-20 CN disclosed
CN-1227248-C Imidazolidine derivatives, their preparation, and their use as antinflamatory agent AVENTIS PHARMA GMBH (DE) 2005-11-16 CN disclosed
CN-1221535-C Spiroimidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them AVENTIS PHARMA GMBH (DE) 2005-10-05 CN disclosed
CN-1496360-A Imidazolidine derivatives, their preparation, and their use as antinflamatory agent ������ҽҩ�¹����޹�˾ 2004-05-12 CN disclosed
CN-1433431-A Interleukin-1 receptor antagonist-like molecules and uses thereof AMGEN INC (US) 2003-07-30 CN disclosed
CN-1356986-A Spiroimidazolidine derivatives, their prepn. their use and pharmaceutical prepns. comprising them AVENTIS PHARMA GMBH (DE) 2002-07-03 CN disclosed