SCHEMBL27520101

SCHEMBL27520101

CC(CCC(O)OCCCN1CCC(c2noc3cc(F)ccc23)CC1)C(=O)C(C)CCC(O)OCCCN1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.62
HTR2A P28223 4/20 0.62
HTR7 P34969 1/20 0.62
HTR1A P08908 3/20 0.61
ADRA2A P08913 2/20 0.61
HTR2C P28335 2/20 0.61
ADRA1A P35348 2/20 0.61
HRH1 P35367 2/20 0.61
HTR6 P50406 2/20 0.61
KCNH2 Q12809 2/20 0.61
ABCB11 O95342 1/20 0.61
CHRM2 P08172 1/20 0.61
CHRM1 P11229 1/20 0.61
ADRA2B P18089 1/20 0.61
ADRA2C P18825 1/20 0.61
DRD1 P21728 1/20 0.61
DRD4 P21917 1/20 0.61
ACHE P22303 1/20 0.61
SLC6A2 P23975 1/20 0.61
SLC6A4 P31645 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545419 0.81 DRD2 (0.76) DRD2HTR2AHTR7KCNH2ACHE
SCHEMBL1545162 0.81 DRD2 (0.76) DRD2HTR2AHTR7KCNH2ACHE
SCHEMBL1545164 0.81 DRD2 (0.76) DRD2HTR2AHTR7KCNH2ACHE
SCHEMBL8714677 0.80 HTR2A (0.62) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL1544927 0.79 HTR1A (0.80) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL22149696 0.79 DRD2 (0.76) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL8523709 0.79 HTR2A (0.62) DRD2HTR2AHTR1AADRA2AHTR2C
Methyl Alcohol SCHEMBL3645347 0.79 DRD2 (0.61) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL1545151 0.79 DRD2 (0.72) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL27523350 0.78 HTR2A (0.65) DRD2HTR2AHTR1AADRA2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1086387-C N- (aryloxyalkyl) heteroarylpiperidines and heteroarylpiperazines, their preparation and their use as pharmaceuticals HOECHST MARION ROUSSEL INC (US) 2002-06-19 CN disclosed
CN-1048037-A N- (aryloxyalkyl) heteroarylpiperidines and heteroarylpiperazines, their preparation and their use as pharmaceuticals HOECHST ROUSSEL PHARMA (US) 1990-12-26 CN disclosed