SCHEMBL8523709

SCHEMBL8523709

COc1ccc(C(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)C(N)=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.62
HTR1A P08908 5/20 0.62
DRD2 P14416 4/20 0.62
ADRA2A P08913 2/20 0.62
HTR2C P28335 2/20 0.62
ADRA1A P35348 2/20 0.62
HRH1 P35367 2/20 0.62
HTR6 P50406 2/20 0.62
KCNH2 Q12809 2/20 0.62
DRD3 P35462 2/20 0.62
ABCB11 O95342 1/20 0.62
CHRM2 P08172 1/20 0.62
CHRM1 P11229 1/20 0.62
ADRA2B P18089 1/20 0.62
ADRA2C P18825 1/20 0.62
DRD1 P21728 1/20 0.62
DRD4 P21917 1/20 0.62
ACHE P22303 1/20 0.62
SLC6A2 P23975 1/20 0.62
SLC6A4 P31645 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8714677 0.90 HTR2A (0.62) HTR2AHTR1ADRD2ADRA2AHTR2C
SCHEMBL27513300 0.81 HTR2A (0.69) HTR2AHTR1ADRD2ADRA2AHTR2C
SCHEMBL1545822 0.80 HTR1A (0.72) HTR2AHTR1ADRD2ADRA2AHTR2C
Anisole SCHEMBL3645349 0.80 DRD2 (0.63) HTR2AHTR1ADRD2ADRA2AHTR2C
SCHEMBL1544927 0.80 HTR1A (0.80) HTR2AHTR1ADRD2ADRA2AHTR2C
SCHEMBL7963611 0.80 HTR6 (0.74) HTR2AHTR1ADRD2HTR2CADRA1A
SCHEMBL8671507 0.80 HTR2A (0.52) HTR2AHTR1ADRD2ADRA2AHTR2C
Hydrochloric Acid SCHEMBL1545292 0.80 HTR1A (0.71) HTR2AHTR1ADRD2ADRA2AHTR2C
SCHEMBL8716361 0.80 HTR1A (0.68) HTR2AHTR1ADRD2ADRA2AHTR2C
SCHEMBL7881728 0.79 ABCB11 (0.76) HTR2AHTR1ADRD2ADRA2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889035-A 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed