SCHEMBL27520459

SCHEMBL27520459

O=C(O)Nc1ccc(CN2CCC(Br)C2=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 1/20 0.46
PKM P14618 2/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
FPR2 P25090 1/20 0.43
LMNA P02545 1/20 0.43
THRB P10828 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
HCRTR1 O43613 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569448 0.82 DRD2 (0.45) TNIKHDAC8KDM4EALDH1A1FPR2
SCHEMBL27485081 0.82 PTGS1 (0.46) HDAC1HDAC8HDAC6KDM4EALDH1A1
SCHEMBL8560030 0.81 TGM2 (0.46) TNIKKDM4EALDH1A1L3MBTL1LMNA
SCHEMBL16874550 0.80 KCNH2 (0.51) LMNA
SCHEMBL8564264 0.79 DDB1 (0.50) HDAC1HDAC8HDAC6ALDH1A1L3MBTL1
SCHEMBL8564268 0.79 DDB1 (0.50) HDAC1HDAC8HDAC6ALDH1A1L3MBTL1
SCHEMBL1542776 0.78 ALDH1A1 (0.49) KDM4EALDH1A1
SCHEMBL8563968 0.78 HDAC8 (0.40) PKMHDAC1HDAC8HDAC6ALDH1A1
SCHEMBL8564966 0.77 ALDH1A1 (0.53) ALDH1A1HTTRAB9A
SCHEMBL8564961 0.77 ALDH1A1 (0.53) ALDH1A1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1150950-A Cephalosporin derivatives HOFFMANN LA ROCHE (CH) 1997-06-04 CN disclosed