SCHEMBL27587725

SCHEMBL27587725

COc1cccc(N(C(N)=O)c2ccc(O)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.50
PARP1 P09874 1/20 0.47
MTNR1A P48039 10/20 0.46
MTNR1B P49286 10/20 0.46
HSD17B2 P37059 2/20 0.44
HSD17B1 P14061 1/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
PTGIR P43119 1/20 0.42
PTGDR Q13258 1/20 0.42
AR P10275 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28382188 0.91 PARP1 (0.56) PARP1MTNR1AMTNR1BHSD17B2HSD17B1
SCHEMBL27515960 0.84 ESR2 (0.52) PARP1CES2CES1
SCHEMBL27495391 0.83 MTNR1B (0.45) PARP1MTNR1AMTNR1BHSD17B2HSD17B1
SCHEMBL27587717 0.80 MTNR1A (0.46) PARP1MTNR1AMTNR1BHSD17B2HSD17B1
SCHEMBL28844152 0.78 TRPM8 (0.56) PARP1MTNR1AMTNR1BCES2CES1
SCHEMBL15779182 0.77 MTNR1A (0.46) PARP1MTNR1AMTNR1BHSD17B2HSD17B1
SCHEMBL3470955 0.77 CA1 (0.55) PARP1CES2CES1
SCHEMBL27296095 0.77 NPSR1 (0.52) ESR1CES2
SCHEMBL22187338 0.77 ESR1 (0.45) ESR1PARP1MTNR1AMTNR1BHSD17B2
SCHEMBL27605653 0.77 CYP3A4 (0.44) ESR1PARP1MTNR1AMTNR1BHSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1539816-A IL-8 receptor antagonists ʷ��˿�������ȳ�ķ���޹�˾ 2004-10-27 CN disclosed