SCHEMBL27622892

SCHEMBL27622892

Cc1ccc(C=Nc2ccc(C(C)(C)C)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.64
CA1 P00915 4/20 0.64
ALDH1A1 P00352 2/20 0.59
TSHR P16473 1/20 0.56
PTGS2 P35354 4/20 0.54
PTGS1 P23219 2/20 0.54
CA9 Q16790 2/20 0.54
CA12 O43570 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12633723 0.86 ALDH1A1 (0.74) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL20186922 0.86 ALDH1A1 (0.74) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL255410 0.86 ALDH1A1 (0.74) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL11588746 0.86 ALDH1A1 (0.74) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL11557679 0.86 ALDH1A1 (0.74) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL29205583 0.84 CA1 (0.62) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL13580880 0.84 CA2 (0.62) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL28964176 0.84 PTGS2 (0.60) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL23219506 0.83 CA1 (0.66) CA2CA1ALDH1A1PTGS2PTGS1
SCHEMBL23219507 0.83 CA1 (0.66) CA2CA1ALDH1A1PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100335468-C Diaryl amidine compound, its production, medicinal composition and use DRUG INST CHINESE ACADEMY OF M (CN) 2007-09-05 CN disclosed
CN-1712398-A Diaryl amidine compound, its production, medicinal composition and use DRUG INST CHINESE ACADEMY OF M (CN) 2005-12-28 CN disclosed