SCHEMBL27639367

SCHEMBL27639367

c1ccc(COc2ccc3cccc(CCc4ccncc4)c3c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.58
ALOX5 P09917 1/20 0.52
CYP3A4 P08684 1/20 0.51
MTNR1A P48039 4/20 0.48
MTNR1B P49286 4/20 0.48
PLAU P00749 1/20 0.48
PLAT P00750 1/20 0.48
F2 P00734 2/20 0.47
KCNH2 Q12809 1/20 0.47
GRIN2B Q13224 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
NPC1 O15118 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15955987 0.78 TRPM8 (0.70) HTR1ALTA4H
SCHEMBL3248265 0.77 MTNR1A (0.66) MTNR1AMTNR1BAKR1B1
SCHEMBL15956138 0.76 TRPM8 (0.57) ABCB1SMN1; SMN2ALDH1A1HPGDHTR1A
SCHEMBL17188139 0.75 ALOX5 (0.56) ALOX5CYP3A4MTNR1AMTNR1BPLAU
SCHEMBL27660097 0.75 ALOX5 (0.56) ALOX5CYP3A4MTNR1AMTNR1BPLAU
SCHEMBL13097042 0.74 LTA4H (0.61) ABCB1F2KCNH2GRIN2BSMN1; SMN2
SCHEMBL4489367 0.74 MRGPRX4 (0.50) ALOX5CYP3A4PLAUPLATSMN1; SMN2
SCHEMBL10606515 0.74 ALOX5 (0.67) ALOX5CYP3A4MTNR1APLAUPLAT
SCHEMBL8783402 0.73 F2 (0.63) ABCB1F2KCNH2GRIN2BSMN1; SMN2
SCHEMBL29227079 0.73 ABCB1 (0.58) ABCB1SMN1; SMN2ALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100455579-C Compounds and compositions as protein kinase inhibitors IRM LLC (BM) 2009-01-28 CN disclosed
CN-1860111-A Compounds and compositions as protein kinase inhibitors IRM LLC (BM) 2006-11-08 CN disclosed