SCHEMBL2766091

SCHEMBL2766091

COc1cc(-c2nc(CN3CCN(Cc4coc(-c5cc(OC)c(OC)c(OC)c5)n4)CC3)co2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.52
DRD4 P21917 4/20 0.52
DRD3 P35462 4/20 0.52
ABCB1 P08183 5/20 0.50
ABCC1 P33527 3/20 0.50
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 3/20 0.45
HPGD P15428 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.44
GAA P10253 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
GLA P06280 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TGFBR1 P36897 1/20 0.41
ACVR1 Q04771 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2764403 0.96 DRD2 (0.49) DRD2DRD4DRD3ABCB1ABCC1
SCHEMBL2764515 0.80 KDM4E (0.50) ALDH1A1KDM4EHPGDL3MBTL1MAPT
SCHEMBL2764253 0.80 KDM4E (0.50) ALDH1A1KDM4EHPGDL3MBTL1MAPT
SCHEMBL3071421 0.77 ABCB1 (0.55) DRD2DRD4DRD3ABCB1ABCC1
SCHEMBL2765382 0.75 TP53 (0.49) ALDH1A1KDM4ETP53MAPTGAA
SCHEMBL2766572 0.74 HTR7 (0.61) DRD2DRD4DRD3ABCB1ABCC1
SCHEMBL5679677 0.73 TP53 (0.47) ALDH1A1KDM4ETP53GAAMEN1
SCHEMBL3087050 0.73 HRH3 (0.57) DRD2DRD4DRD3ABCB1ABCC1
SCHEMBL5681214 0.72 TP53 (0.52) ALDH1A1KDM4ETP53GAAMEN1
SCHEMBL2767252 0.72 KDM4E (0.49) ALDH1A1KDM4ETP53GAAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1400515-B1 CYCLIC DIAMINE COMPOUND HAVING FIVE-MEMBERED CYCLIC GROUP KOWA CO (JP) 2010-04-14 EP disclosed
EP-1400515-A1 CYCLIC DIAMINE COMPOUND HAVING FIVE-MEMBERED CYCLIC GROUP Kowa Co., Ltd. (JP) 2004-03-24 EP disclosed
US-6472386-B1 Cyclic diamine compound with 5-membered ring groups KOWA CO., LTD. (JP) 2002-10-29 US disclosed