SCHEMBL27670545

SCHEMBL27670545

COC(=O)Cc1cccc(N2CCNC2=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSG P08311 2/20 0.48
CMA1 P23946 2/20 0.48
TSHR P16473 2/20 0.45
SLC7A5 Q01650 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
DRD2 P14416 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTR7 P34969 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2B P41595 1/20 0.42
KCNH2 Q12809 1/20 0.42
ALDH1A1 P00352 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5727052 0.84 HSD17B10 (0.49) CTSGCMA1TSHRKCNH2ALDH1A1
SCHEMBL2878333 0.84 ITGB3 (0.48) CYP1A2CYP3A4HTR1ACYP2D6CYP2C9
SCHEMBL27670559 0.81 ALDH1A1 (0.46) CTSGCMA1TSHRHTR7KCNH2
SCHEMBL27765009 0.79 ALOX5 (0.52) CMA1CYP1A2CYP3A4HTR1ACYP2D6
SCHEMBL4577325 0.79 ADRB1 (0.55) CTSGCMA1SLC7A5CYP1A2CYP3A4
SCHEMBL13853443 0.78 DDB1 (0.51) CYP1A2CYP3A4HTR1ACYP2D6CYP2C9
SCHEMBL132460 0.77 GAA (0.55) CTSGCMA1TSHRCYP1A2CYP2D6
SCHEMBL15709650 0.77 PRMT6 (0.56) CTSGCMA1TSHRSLC7A5ALDH1A1
SCHEMBL2885321 0.77 HTR1A (0.48) CYP1A2CYP3A4HTR1ACYP2D6CYP2C9
SCHEMBL15709874 0.77 MAPT (0.53) CTSGCMA1TSHRSLC7A5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100441571-C Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors GLAXO GROUP LTD (GB) 2008-12-10 CN disclosed
CN-1852896-A Quinoline and quinazoline derivatives having affinity for 5HT 1-type receptors GLAXO GROUP LTD (GB) 2006-10-25 CN disclosed