SCHEMBL27675114

SCHEMBL27675114

COc1cc(OC)c(-c2ccccc2NC(=O)n2cc(C(=O)O)c(=O)c3ccccc32)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
ALDH1A1 P00352 4/20 0.36
HTT P42858 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 5/20 0.36
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
POLB P06746 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
CHEK1 O14757 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675229 0.86 KDM4E (0.45) CHRM1L3MBTL1MEN1KMT2AALDH1A1
SCHEMBL27693793 0.81 KMT2A (0.51) CHRM1MEN1KMT2ARAB9AKDM4E
SCHEMBL27991300 0.79 KDM4E (0.43) CHRM1L3MBTL1MEN1KMT2AALDH1A1
SCHEMBL27693506 0.78 CREBBP (0.49) CHRM1L3MBTL1KMT2AALDH1A1RAB9A
SCHEMBL27675331 0.78 CFD (0.41) S1PR1S1PR3ALDH1A1KDM4EHPGD
SCHEMBL27693557 0.77 LMNA (0.40) CHRM1L3MBTL1ALDH1A1RAB9AKDM4E
SCHEMBL27920808 0.77 KDM4E (0.41) L3MBTL1S1PR1S1PR3MEN1KMT2A
SCHEMBL27675161 0.77 POLB (0.43) CHRM1L3MBTL1MEN1KMT2AALDH1A1
SCHEMBL27693660 0.76 POLB (0.44) CHRM1MEN1KMT2AALDH1A1KDM4E
SCHEMBL27675213 0.75 HTT (0.46) CHRM1S1PR1S1PR3ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed